SCHEMBL12677220

SCHEMBL12677220

COc1cc(N)c(I)cc1C(C)=O

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.47
GAA P10253 1/20 0.46
HTT P42858 2/20 0.46
ACHE P22303 3/20 0.44
HTR4 Q13639 3/20 0.44
CA9 Q16790 1/20 0.43
ALDH1A1 P00352 2/20 0.42
CYP3A4 P08684 2/20 0.42
LMNA P02545 2/20 0.40
CFTR P13569 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
NQO2 P16083 1/20 0.38
RAB9A P51151 1/20 0.37
TSHR P16473 1/20 0.37
POLB P06746 1/20 0.37
APP P05067 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7801336 0.86 ALDH1A1 (0.54) KDM4EGAAHTTACHEHTR4
SCHEMBL2596444 0.84 GAA (0.66) KDM4EGAAHTTACHEHTR4
SCHEMBL1219388 0.83 CYP3A4 (0.50) HTTACHECA9ALDH1A1CYP3A4
SCHEMBL24106157 0.80 HTT (0.61) KDM4EGAAHTTACHECA9
SCHEMBL6371675 0.79 CYP3A4 (0.55) KDM4EGAAHTTCA9ALDH1A1
SCHEMBL16400171 0.79 HTR4 (0.48) KDM4EGAAACHEHTR4ALDH1A1
SCHEMBL7351910 0.79 GAA (0.73) GAAHTR4ALDH1A1CYP3A4LMNA
SCHEMBL20630769 0.78 HTT (0.68) KDM4EHTTCA9ALDH1A1CYP3A4
SCHEMBL23015575 0.78 HTR4 (0.55) KDM4EGAAACHEHTR4ALDH1A1
SCHEMBL24106211 0.77 TNFSF11 (0.51) HTTCA9CYP3A4LMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2316469-A1 Delivery system and methods for protecting and administering dextroamphetamine Shire LLC (US) 2011-05-04 EP disclosed