SCHEMBL12699666

SCHEMBL12699666

c1ccc(-c2ccc3c4ccccc4n(-c4ccc5cc(-n6c7ccccc7c7ccc(-c8ccccc8)cc76)ccc5c4)c3c2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.48
ATM Q13315 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
HDAC4 P56524 1/20 0.40
RXRA P19793 1/20 0.40
RXRB P28702 1/20 0.40
ESR1 P03372 3/20 0.40
ESR2 Q92731 3/20 0.40
LDHA P00338 1/20 0.39
F2 P00734 1/20 0.37
F10 P00742 1/20 0.37
PRSS1 P07477 1/20 0.37
HTR6 P50406 1/20 0.37
FGFR1 P11362 1/20 0.36
KMT2A Q03164 2/20 0.35
MAOB P27338 1/20 0.35
MAPK9 P45984 1/20 0.35
MAPK10 P53779 1/20 0.35
MEN1 O00255 1/20 0.35
HSP90AA1 P07900 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19500801 0.97 L3MBTL1 (0.50) KDM4EATML3MBTL1HDAC4RXRA
SCHEMBL21709230 0.97 KDM4E (0.46) KDM4EATML3MBTL1HDAC4RXRA
SCHEMBL19500800 0.95 KDM4E (0.44) KDM4EATML3MBTL1HDAC4RXRA
SCHEMBL19036992 0.95 KDM4E (0.49) KDM4EATML3MBTL1HDAC4RXRA
SCHEMBL19500798 0.95 KDM4E (0.49) KDM4EATML3MBTL1HDAC4RXRA
SCHEMBL19500797 0.95 L3MBTL1 (0.53) KDM4EATML3MBTL1HDAC4RXRA
SCHEMBL19500802 0.94 ATM (0.47) KDM4EATML3MBTL1HDAC4RXRA
SCHEMBL19500799 0.94 KDM4E (0.44) KDM4EATML3MBTL1HDAC4RXRA
SCHEMBL19131225 0.93 ATM (0.46) KDM4EATML3MBTL1HDAC4RXRA
SCHEMBL19500787 0.93 KDM4E (0.46) KDM4EATML3MBTL1HDAC4RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2627730-B1 FORMULATIONS FOR ORGANIC ELECTROLUMINESCENCE DEVICES MERCK PATENT GMBH (DE) 2020-05-06 EP disclosed
EP-2627732-B1 MATERIALS FOR ORGANIC ELECTROLUMINESCENCE DEVICES MERCK PATENT GMBH (DE) 2017-12-20 EP disclosed
US-9653687-B2 Materials for organic electroluminescent devices MERCK PATENT GMBH (DE) 2017-05-16 US disclosed
US-9653687-B2 Materials for organic electroluminescent devices MERCK PATENT GMBH (DE) 2017-05-16 US disclosed
EP-2787053-A1 Polymeric materials Merck Patent GmbH (DE) 2014-10-08 EP disclosed
US-8786181-B2 Materials for organic electroluminescent devices MERCK PATENT GMBH (DE) 2014-07-22 US disclosed
US-8786181-B2 Materials for organic electroluminescent devices MERCK PATENT GMBH (DE) 2014-07-22 US disclosed
US-20130228767-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK 2013-09-05 US disclosed
US-20130228767-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK 2013-09-05 US disclosed
US-20130207095-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES Fraunhofer-Gesellschaft Forderung E.V. (DE) 2013-08-15 US disclosed
US-20130207095-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES Fraunhofer-Gesellschaft Forderung E.V. (DE) 2013-08-15 US disclosed
US-20130200357-A1 FORMULATIONS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2013-08-08 US disclosed
US-20130200357-A1 FORMULATIONS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2013-08-08 US disclosed
US-8343637-B2 Carbazole derivatives for organic electroluminescent devices MERCK PATENT GMBH (DE) 2013-01-01 US disclosed
US-8343637-B2 Carbazole derivatives for organic electroluminescent devices MERCK PATENT GMBH (DE) 2013-01-01 US disclosed
WO-2012048900-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENCE DEVICES FRAUNHOFER-GESELLSCHAFT ZUR FÖRDERUNG DER ANGEWANDTEN FORSCHUNG E.V. . (DE) 2012-04-19 WO disclosed
EP-2102309-B1 CARBAZOLE DERIVATIVES FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2010-06-30 EP disclosed
US-20090302752-A1 CARBAZOLE DERIVATIVES FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2009-12-10 US disclosed
US-20090302752-A1 CARBAZOLE DERIVATIVES FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2009-12-10 US disclosed
WO-2008086851-A1 CARBAZOLE DERIVATIVES FOR ORGANC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2008-07-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090302752-A1 CARBAZOLE DERIVATIVES FOR ORGANIC ELECTROLUMINESCENT DEVICES PIEZO1, CACNA2D1, CYCS KDM4E 3257/4885ATM 3616/4885L3MBTL1 3911/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.