SCHEMBL12712312

SCHEMBL12712312

C/C=N\C(=C(/C)Cl)c1cc(C)nc2c(OCc3c(Cl)ccnc3CNC(=O)C(C)C)cccc12

nearest known ligand 0.53

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BDKRB2 P30411 20/20 0.53
CYP3A4 P08684 2/20 0.53
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13093092 0.93 BDKRB2 (0.61) BDKRB2CYP3A4CYP2C19
SCHEMBL12711415 0.93 BDKRB2 (0.47) BDKRB2CYP3A4
SCHEMBL12711930 0.93 BDKRB2 (0.46) BDKRB2CYP3A4CYP2C19
SCHEMBL12711445 0.89 BDKRB2 (0.41) BDKRB2CYP3A4CYP2C19
SCHEMBL12711446 0.89 BDKRB2 (0.51) BDKRB2CYP3A4CYP2C19
SCHEMBL12711939 0.87 BDKRB2 (0.62) BDKRB2CYP3A4
SCHEMBL12711396 0.87 BDKRB2 (0.62) BDKRB2CYP3A4CYP2C19
SCHEMBL13093084 0.86 BDKRB2 (0.54) BDKRB2CYP3A4CYP2C19
SCHEMBL13093152 0.85 BDKRB2 (0.48) BDKRB2CYP3A4
SCHEMBL13092925 0.85 BDKRB2 (0.46) BDKRB2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2305668-A1 8-oxy-quinoline derivatives as bradykinin B2 receptor modulators Jerini AG (DE) 2011-04-06 EP disclosed
WO-2008116620-A1 8-OXY-QUINOLINE DERIVATIVES AS BRADYKININ B2 RECEPTOR MODULATORS JERINI AG (DE) 2008-10-02 WO disclosed