SCHEMBL12778304

SCHEMBL12778304

Cc1ccnc2[nH]c(I)nc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 2/20 0.38
CCR5 P51681 2/20 0.38
CCR8 P51685 2/20 0.38
GSK3A P49840 6/20 0.37
GSK3B P49841 6/20 0.37
CCNB2 O95067 5/20 0.37
CDK1 P06493 5/20 0.37
CCNB1 P14635 5/20 0.37
CCNB3 Q8WWL7 5/20 0.37
CDK5 Q00535 4/20 0.37
CDK5R1 Q15078 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.33
NOS3 P29474 2/20 0.32
NOS2 P35228 2/20 0.32
CBFB Q13951 1/20 0.32
HTR1A P08908 1/20 0.32
ADRA1D P25100 1/20 0.32
ADRA1A P35348 1/20 0.32
ADRA1B P35368 1/20 0.32
MAPK8 P45983 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1665498 0.80 PARP1 (0.42) CCR1CCR5CCR8GSK3AGSK3B
SCHEMBL12778306 0.77 TSHR (0.38) GSK3AGSK3BCCNB2CDK1CCNB1
SCHEMBL12777919 0.77 MAPK14 (0.34) GSK3AGSK3BCCNB2CDK1CCNB1
SCHEMBL21620891 0.77 NOS3 (0.41) CCR1CCR5CCR8GSK3AGSK3B
SCHEMBL21620456 0.77 CCNB2 (0.40) CCR1CCR5CCR8GSK3AGSK3B
SCHEMBL8558723 0.77 PSMD14 (0.38) CCR1CCR5CCR8GSK3AGSK3B
SCHEMBL12778307 0.77 CDK5 (0.39) GSK3AGSK3BCCNB2CDK1CCNB1
SCHEMBL14336690 0.74 CCR1 (0.35) CCR1CCR5CCR8GSK3AGSK3B
SCHEMBL4370028 0.74 ADORA1 (0.41) CCR1CCR5CCR8GSK3AGSK3B
SCHEMBL15925243 0.74 DAO (0.40) AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011050160-A1 PHARMACEUTICALS, COMPOSITIONS AND METHODS OF MAKING AND USING THE SAME BIOGEN IDEC MA INC. (US) 2011-04-28 WO disclosed