SCHEMBL12801015

SCHEMBL12801015

Cc1noc(C)c1-c1c(-c2ccc(O)cc2)c(C(F)(F)F)n(C)c1N

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 2/20 0.45
BRD4 O60885 13/20 0.39
BRD2 P25440 2/20 0.38
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
BRD3 Q15059 1/20 0.36
ERN1 O75460 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
JAK2 O60674 1/20 0.35
USP7 Q93009 1/20 0.34
CREBBP Q92793 1/20 0.34
TDO2 P48775 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1670795 0.83 AR (0.44) MLYCDBRD4BRD2ESR1ESR2
SCHEMBL12800382 0.81 MLYCD (0.42) MLYCDBRD4BRD2BRD3ERN1
SCHEMBL12801001 0.78 BRD4 (0.39) MLYCDBRD4BRD2BRD3ERN1
SCHEMBL12801014 0.77 ERN1 (0.41) MLYCDBRD4BRD2BRD3ERN1
SCHEMBL12800390 0.75 BRD4 (0.43) MLYCDBRD4BRD2BRD3ERN1
SCHEMBL12362813 0.74 BRD4 (0.66) MLYCDBRD4BRD2ERN1CREBBP
SCHEMBL12808114 0.74 BRD4 (0.45) MLYCDBRD4BRD2BRD3ERN1
Hydrochloric Acid SCHEMBL23174957 0.73 BRD4 (0.63) MLYCDBRD4BRD2ERN1CREBBP
SCHEMBL12800997 0.72 BRD4 (0.42) MLYCDBRD4BRD2ERN1JAK2
SCHEMBL10200524 0.68 MAP4K4 (0.56) MLYCDBRD4BRD2JAK2USP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011042477-A1 SUBSTITUTED PYRROLES AND IMIDAZOLES AS ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO disclosed