SCHEMBL12801355

SCHEMBL12801355

Nc1cc(-c2ccnc(Nc3cccc(N4CCOCC4)c3)n2)ccc1OC1CCOCC1

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CAMK2D Q13557 1/20 0.60
JAK2 O60674 8/20 0.59
TBK1 Q9UHD2 5/20 0.59
JAK3 P52333 2/20 0.53
MAPK8 P45983 2/20 0.51
MAPK10 P53779 2/20 0.51
PLK4 O00444 1/20 0.51
SMG1 Q96Q15 4/20 0.51
CDK1 P06493 2/20 0.51
CDK2 P24941 2/20 0.51
MTOR P42345 1/20 0.51
IKBKE Q14164 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12801662 0.91 JAK2 (0.68) JAK2TBK1JAK3IKBKE
SCHEMBL12801583 0.90 IKBKE (0.56) CAMK2DJAK2TBK1IKBKE
SCHEMBL12521832 0.90 TBK1 (0.53) CAMK2DJAK2TBK1JAK3IKBKE
SCHEMBL1667748 0.88 TBK1 (0.77) JAK2TBK1IKBKE
SCHEMBL12801576 0.87 JAK2 (0.65) JAK2TBK1JAK3
SCHEMBL12800953 0.87 ABL1 (0.56) CAMK2DJAK2TBK1IKBKE
SCHEMBL12801266 0.87 IKBKE (0.54) TBK1IKBKE
SCHEMBL12801672 0.86 TBK1 (0.57) JAK2TBK1SMG1IKBKE
SCHEMBL13467176 0.86 IKBKE (0.56) JAK2TBK1JAK3IKBKE
SCHEMBL12801307 0.86 JAK2 (0.66) JAK2TBK1JAK3MAPK8PLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed