SCHEMBL12801672

SCHEMBL12801672

Nc1cc(-c2ccnc(Nc3ccccc3)n2)ccc1OC1CCOCC1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 17/20 0.57
IKBKE Q14164 16/20 0.57
SMG1 Q96Q15 1/20 0.53
IKBKB O14920 1/20 0.52
JAK2 O60674 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12801583 0.92 IKBKE (0.56) TBK1IKBKEJAK2
SCHEMBL12801120 0.92 IKBKE (0.57) TBK1IKBKEJAK2
SCHEMBL12801266 0.91 IKBKE (0.54) TBK1IKBKE
SCHEMBL12801135 0.90 IKBKE (0.56) TBK1IKBKEJAK2
SCHEMBL12801392 0.90 IKBKE (0.56) TBK1IKBKEJAK2
SCHEMBL12522270 0.89 IKBKE (0.55) TBK1IKBKEJAK2
SCHEMBL12801215 0.89 IKBKE (0.54) TBK1IKBKEJAK2
SCHEMBL12800939 0.89 IKBKE (0.54) TBK1IKBKEJAK2
SCHEMBL12801677 0.88 ABL1 (0.53) TBK1IKBKE
SCHEMBL12801078 0.88 IKBKE (0.61) TBK1IKBKEJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed