SCHEMBL12801583

SCHEMBL12801583

Nc1cccc(Nc2nccc(-c3ccc(OC4CCOCC4)c(N)c3)n2)c1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IKBKE Q14164 15/20 0.56
TBK1 Q9UHD2 15/20 0.56
CDK5 Q00535 1/20 0.55
ABL1 P00519 2/20 0.54
BCR P11274 2/20 0.54
SRC P12931 2/20 0.54
JAK2 O60674 1/20 0.53
EGFR P00533 1/20 0.53
PRKACA P17612 1/20 0.53
PRKACG P22612 1/20 0.53
PRKACB P22694 1/20 0.53
CAMK2D Q13557 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12801266 0.93 IKBKE (0.54) IKBKETBK1CDK5
SCHEMBL12801672 0.92 TBK1 (0.57) IKBKETBK1JAK2
SCHEMBL12801355 0.90 CAMK2D (0.60) IKBKETBK1JAK2CAMK2D
SCHEMBL12801120 0.90 IKBKE (0.57) IKBKETBK1JAK2
SCHEMBL12801677 0.90 ABL1 (0.53) IKBKETBK1ABL1BCRSRC
SCHEMBL12801655 0.89 IKBKE (0.60) IKBKETBK1
SCHEMBL12800406 0.89 JAK2 (0.56) IKBKETBK1CDK5JAK2
SCHEMBL12801714 0.89 ABL1 (0.55) IKBKETBK1ABL1BCRSRC
SCHEMBL1667274 0.88 TBK1 (0.73) IKBKETBK1
SCHEMBL12801719 0.88 JAK2 (0.55) IKBKETBK1JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed