SCHEMBL12801392

SCHEMBL12801392

Nc1cc(-c2ccnc(Nc3ccc(-c4ccncc4)cc3)n2)ccc1OC1CCOCC1

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
IKBKE Q14164 19/20 0.56
TBK1 Q9UHD2 19/20 0.56
JAK2 O60674 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12801120 0.92 IKBKE (0.57) IKBKETBK1JAK2
SCHEMBL12801677 0.92 ABL1 (0.53) IKBKETBK1
SCHEMBL12522270 0.91 IKBKE (0.55) IKBKETBK1JAK2
SCHEMBL12801135 0.90 IKBKE (0.56) IKBKETBK1JAK2
SCHEMBL12801082 0.90 TBK1 (0.54) IKBKETBK1JAK2
SCHEMBL12801672 0.90 TBK1 (0.57) IKBKETBK1JAK2
SCHEMBL12800939 0.89 IKBKE (0.54) IKBKETBK1JAK2
SCHEMBL12801215 0.89 IKBKE (0.54) IKBKETBK1JAK2
SCHEMBL12801078 0.88 IKBKE (0.61) IKBKETBK1JAK2
SCHEMBL12801662 0.88 JAK2 (0.68) IKBKETBK1JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed