SCHEMBL12801677

SCHEMBL12801677

Nc1cc(-c2ccnc(Nc3cccc(-c4ccncc4)c3)n2)ccc1OC1CCOCC1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 2/20 0.53
BCR P11274 2/20 0.53
SRC P12931 2/20 0.53
IKBKE Q14164 16/20 0.52
TBK1 Q9UHD2 16/20 0.52
SYK P43405 2/20 0.47
EGFR P00533 1/20 0.46
PRKACA P17612 1/20 0.46
PRKACG P22612 1/20 0.46
PRKACB P22694 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12801714 0.92 ABL1 (0.55) ABL1BCRSRCIKBKETBK1
SCHEMBL12801392 0.92 IKBKE (0.56) IKBKETBK1
SCHEMBL12801583 0.90 IKBKE (0.56) ABL1BCRSRCIKBKETBK1
SCHEMBL12801266 0.88 IKBKE (0.54) IKBKETBK1
SCHEMBL12801672 0.88 TBK1 (0.57) IKBKETBK1
SCHEMBL1667827 0.87 IKBKE (0.70) IKBKETBK1
SCHEMBL12522270 0.87 IKBKE (0.55) ABL1BCRSRCIKBKETBK1
SCHEMBL12800406 0.85 JAK2 (0.56) IKBKETBK1
SCHEMBL12801655 0.85 IKBKE (0.60) IKBKETBK1
SCHEMBL12801355 0.84 CAMK2D (0.60) IKBKETBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed