SCHEMBL12801517

SCHEMBL12801517

CC(C)COc1ccc(-c2ccnc(Cl)n2)cc1N

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
XDH P47989 6/20 0.57
AAK1 Q2M2I8 7/20 0.46
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
KMO O15229 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12801634 0.82 KMO (0.50) AAK1ALDH1A1KMO
SCHEMBL12448384 0.81 AAK1 (0.61) XDHAAK1
SCHEMBL12801515 0.79 KMO (0.56) XDHKMO
SCHEMBL21508531 0.77 AAK1 (0.44) AAK1KMO
SCHEMBL12801516 0.76 DHFR (0.42) XDHAAK1KMO
SCHEMBL21508770 0.76 AAK1 (0.50) XDHAAK1KMO
SCHEMBL12801571 0.76 KMO (0.51) ALDH1A1KMO
SCHEMBL20446923 0.74 AAK1 (0.56) AAK1KMO
SCHEMBL21508530 0.73 AAK1 (0.58) XDHAAK1
SCHEMBL21508296 0.73 AAK1 (0.58) XDHAAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed