SCHEMBL12801516

SCHEMBL12801516

CC1(COc2ccc(-c3ccnc(Cl)n3)cc2N)COC1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.42
DCPS Q96C86 1/20 0.42
IRAK4 Q9NWZ3 1/20 0.38
FFAR1 O14842 1/20 0.38
BACE1 P56817 4/20 0.37
AAK1 Q2M2I8 3/20 0.36
CHEK1 O14757 1/20 0.36
CHEK2 O96017 1/20 0.36
AKT1 P31749 1/20 0.36
KMO O15229 3/20 0.35
JAK2 O60674 1/20 0.35
TBK1 Q9UHD2 1/20 0.35
GRM2 Q14416 1/20 0.35
XDH P47989 1/20 0.34
CNR2 P34972 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12448386 0.84 TBK1 (0.50) AAK1CHEK1CHEK2AKT1JAK2
SCHEMBL12801634 0.77 KMO (0.50) AAK1KMOJAK2
SCHEMBL12801517 0.76 XDH (0.57) AAK1KMOXDH
SCHEMBL12801129 0.76 JAK2 (0.69) IRAK4AAK1CHEK1CHEK2AKT1
SCHEMBL12801515 0.75 KMO (0.56) KMOXDH
SCHEMBL12801571 0.73 KMO (0.51) KMO
SCHEMBL12801501 0.73 KMO (0.47) KMOTBK1
SCHEMBL19175491 0.69 DHFR (0.43) DHFRDCPSIRAK4BACE1CHEK1
SCHEMBL25257064 0.68 NOS3 (0.49) DHFRDCPSIRAK4BACE1
SCHEMBL12408680 0.67 MEN1 (0.61) KMOJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed