SCHEMBL12801719

SCHEMBL12801719

CC(=O)Nc1cccc(Nc2nccc(-c3ccc(OC4CCOCC4)c(N)c3)n2)c1

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 8/20 0.55
IKBKE Q14164 8/20 0.54
TBK1 Q9UHD2 8/20 0.54
PLK1 P53350 1/20 0.52
IKBKB O14920 1/20 0.49
JAK3 P52333 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
LRRK2 Q5S007 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12801132 0.91 IKBKE (0.52) JAK2IKBKETBK1
SCHEMBL12801721 0.90 IKBKE (0.51) JAK2IKBKETBK1JAK3
SCHEMBL12800938 0.90 TBK1 (0.51) JAK2IKBKETBK1
SCHEMBL12800945 0.90 IKBKE (0.51) JAK2IKBKETBK1JAK3
SCHEMBL12800943 0.89 IKBKE (0.51) JAK2IKBKETBK1JAK3
SCHEMBL12801648 0.88 IKBKE (0.51) JAK2IKBKETBK1JAK3HDAC1
SCHEMBL1667605 0.88 IKBKE (0.68) IKBKETBK1
SCHEMBL12801583 0.88 IKBKE (0.56) JAK2IKBKETBK1
SCHEMBL12801371 0.88 IKBKE (0.49) JAK2IKBKETBK1JAK3
SCHEMBL12801140 0.87 IKBKE (0.50) JAK2IKBKETBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed