SCHEMBL1280508

SCHEMBL1280508

C=C(C(=O)OC)C(O)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 9/20 0.46
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
SLC6A2 P23975 2/20 0.42
SLC6A4 P31645 2/20 0.42
CASP1 P29466 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1280792 0.87 S1PR3 (0.39) CASP1
SCHEMBL1279942 0.87 MDM2 (0.42) SLC6A3ALDH1A1HTTSMN1; SMN2SLC6A2
SCHEMBL23701224 0.82 MAPT (0.45) ALDH1A1LMNAHTTSMN1; SMN2HPGD
SCHEMBL20048220 0.82 HPGD (0.43) ALDH1A1LMNASMN1; SMN2CASP1HPGD
SCHEMBL18987962 0.81 PDE2A (0.43)
SCHEMBL19021492 0.81 PDE2A (0.43)
SCHEMBL1566492 0.80 SLC6A3 (0.57) SLC6A3ALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL1566494 0.80 SLC6A3 (0.57) SLC6A3ALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL12469122 0.80 KEAP1 (0.42) SLC6A3ALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL15965560 0.77 HPGD (0.44) ALDH1A1LMNASMN1; SMN2CASP1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8722662-B2 Heterocyclic compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2014-05-13 US disclosed
US-20130267494-A1 1,4-OXAZEPANE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-10-10 US disclosed
US-20120088748-A1 HETEROCYCLIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-04-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130267494-A1 1,4-OXAZEPANE DERIVATIVES MAOB, SLC6A4, SLC6A2 SLC6A3 6/4885ALDH1A1 170/4885LMNA 4129/4885
US-20120088748-A1 HETEROCYCLIC COMPOUNDS SLC6A2, MAOB, MAOA SLC6A3 4/4885ALDH1A1 230/4885LMNA 3367/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.