SCHEMBL12809571

SCHEMBL12809571

CCCCCCCCc1ccc2[nH]cc(CNC)c2c1

nearest known ligand 0.70

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 10/20 0.70
HTR1D P28221 9/20 0.70
HTR1B P28222 9/20 0.70
TRPV1 Q8NER1 3/20 0.47
MAPT P10636 2/20 0.46
MAPK1 P28482 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
KDM4E B2RXH2 1/20 0.46
TP53 P04637 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
HTR2A P28223 1/20 0.46
CYP2C19 P33261 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
MPO P05164 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14975308 0.82 HTR1A (1.00) HTR1AHTR1DHTR1BMAPTMAPK1
SCHEMBL5461625 0.82 HTR1A (0.71) HTR1AHTR1DHTR1BTRPV1MAPT
SCHEMBL8920992 0.81 HTR1A (0.97) HTR1AHTR1DHTR1BMAPTMAPK1
SCHEMBL29018529 0.80 HTR1A (0.78) HTR1AHTR1DHTR1BMAPTMAPK1
SCHEMBL10778563 0.80 HTR1A (0.74) HTR1AHTR1DHTR1BTRPV1MPO
SCHEMBL28267254 0.78 HTR1A (0.66) HTR1AHTR1DHTR1BTRPV1MAPT
SCHEMBL5471393 0.77 HTR1A (0.70) HTR1AHTR1DHTR1BTRPV1CYP2D6
SCHEMBL11290643 0.76 HTR1A (0.72) HTR1AHTR1DHTR1BMAPTMAPK1
SCHEMBL13964396 0.75 HTR1A (0.66) HTR1AHTR1DHTR1BHTR2AMPO
SCHEMBL14692901 0.74 HTR1D (0.72) HTR1AHTR1DHTR1BMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2298790-A1 Daptomycin analogs as antibacterial agents Cubist Pharmaceuticals, Inc. (US) 2011-03-23 EP disclosed
EP-2295444-A2 Lipopeptides as antibacterial agents Cubist Pharmaceutical Inc. (US) 2011-03-16 EP disclosed