SCHEMBL12809588

SCHEMBL12809588

CC(C)(C)n1ncc(C(=O)N[C@H]2CCC3CC4CC(C3)C2C4)c1-n1cccn1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 4/20 0.39
HCRTR1 O43613 6/20 0.36
HSD17B10 Q99714 2/20 0.34
CHRM1 P11229 5/20 0.34
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
LMNA P02545 1/20 0.32
TYK2 P29597 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12809751 1.00 HSD11B1 (0.39) HSD11B1HCRTR1HSD17B10CHRM1KDM4E
SCHEMBL12809700 0.87 HSD11B1 (0.41) HSD11B1HCRTR1HSD17B10CHRM1KDM4E
SCHEMBL14412768 0.87 HSD11B1 (0.41) HSD11B1HCRTR1HSD17B10CHRM1KDM4E
SCHEMBL14413253 0.86 HSD11B1 (0.43) HSD11B1HCRTR1
SCHEMBL12809781 0.85 HSD11B1 (0.41) HSD11B1HCRTR1HSD17B10CHRM1
SCHEMBL14412571 0.85 HSD11B1 (0.43) HSD11B1HCRTR1
SCHEMBL1407021 0.85 HSD11B1 (0.54) HSD11B1LMNA
SCHEMBL12809780 0.84 LMNA (0.36) HSD11B1HSD17B10KDM4EALDH1A1HPGD
SCHEMBL12809589 0.84 HSD11B1 (0.34) HSD11B1HSD17B10KDM4EALDH1A1HPGD
SCHEMBL12809752 0.83 CNR2 (0.35) HSD11B1HSD17B10LMNATYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2295411-A1 Pyrazoles as 11-beta-hsd-1 F. Hoffmann-La Roche AG (CH) 2011-03-16 EP disclosed