SCHEMBL12814432

SCHEMBL12814432

COc1ccc(-c2cccc3[nH]c(S)nc23)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.46
PLA2G2A P14555 1/20 0.46
ALOX15 P16050 1/20 0.46
PTGS2 P35354 1/20 0.46
AURKA O14965 1/20 0.46
KDM4E B2RXH2 2/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
ALDH1A1 P00352 1/20 0.46
PKM P14618 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ENPP1 P22413 2/20 0.44
MAPT P10636 2/20 0.43
CASP3 P42574 1/20 0.43
SENP8 Q96LD8 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
SENP6 Q9GZR1 1/20 0.43
ABL1 P00519 1/20 0.41
ABCB1 P08183 1/20 0.41
BCR P11274 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17740425 0.82 ENPP1 (0.46) PARP1PLA2G2AALOX15PTGS2AURKA
SCHEMBL2010618 0.81 CNR2 (0.48) PARP1
SCHEMBL8814866 0.80 KDM4E (0.61) PARP1PLA2G2AALOX15PTGS2AURKA
SCHEMBL8818573 0.78 MGAM (0.60) PARP1PLA2G2AALOX15PTGS2AURKA
SCHEMBL716477 0.74 CBFB (0.54) PARP1ALOX15AURKANPC1RAB9A
SCHEMBL14823682 0.72 NPC1 (0.39) PARP1PLA2G2AALOX15PTGS2AURKA
SCHEMBL3187259 0.71 ABL1 (0.57) PTGS2NPC1RAB9ASMN1; SMN2ENPP1
SCHEMBL29878398 0.71 ENPP1 (0.44) NPC1RAB9AALDH1A1SMN1; SMN2ENPP1
SCHEMBL8816887 0.70 PARP1 (0.53) PARP1PLA2G2AALOX15PTGS2AURKA
SCHEMBL8814869 0.70 PARP1 (0.62) PARP1AURKAKDM4ENPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2691095-A2 IMIDAZOLYL AMIDE COMPOUNDS AND USES RELATED THERETO Emory University (US) 2014-02-05 EP disclosed
WO-2012135296-A2 IMIDAZOLYL AMIDE COMPOUNDS AND USES RELATED THERETO EMORY UNIVERSITY (US) 2012-10-04 WO disclosed