SCHEMBL12825331

SCHEMBL12825331

O=C(O)c1ccc(NC(=O)c2cc(Cl)c(O)c(Cl)c2)nc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 2/20 0.64
GCK P35557 10/20 0.55
RAB9A P51151 4/20 0.53
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
DEGS1 O15121 2/20 0.51
TP53 P04637 3/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
NPC1 O15118 2/20 0.51
CYP1A2 P05177 2/20 0.51
CYP2D6 P10635 2/20 0.51
CYP2C19 P33261 2/20 0.51
CYP3A4 P08684 1/20 0.51
ALOX15 P16050 1/20 0.51
RARA P10276 2/20 0.50
RARB P10826 2/20 0.50
RARG P13631 2/20 0.50
TTR P02766 1/20 0.50
MAPT P10636 1/20 0.49
TSHR P16473 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5239506 0.85 HCAR3 (0.68) HCAR3GCKRAB9AMEN1KMT2A
SCHEMBL9944094 0.84 HCAR3 (0.58) HCAR3GCKRAB9AMEN1KMT2A
SCHEMBL27451977 0.84 HCAR3 (0.69) HCAR3GCKDEGS1RARARARB
SCHEMBL1459281 0.82 RAB9A (0.62) HCAR3GCKRAB9AMEN1KMT2A
SCHEMBL9944145 0.80 MEN1 (0.67) HCAR3GCKRAB9AMEN1KMT2A
SCHEMBL2664544 0.79 HCAR3 (1.00) HCAR3GCKRAB9AMEN1KMT2A
SCHEMBL5236720 0.78 HCAR3 (0.66) HCAR3GCKRAB9AMEN1KMT2A
SCHEMBL5233651 0.78 HCAR3 (0.57) HCAR3GCKRAB9AMEN1KMT2A
SCHEMBL31586306 0.78 HCAR3 (0.57) HCAR3GCKRAB9AMEN1KMT2A
SCHEMBL5237722 0.78 ALDH1A1 (0.58) HCAR3GCKRAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011027106-A1 THERAPEUTIC ARYL-AM I DO-ARYL COMPOUNDS AND THEIR USE KING'S COLLEGE LONDON (GB) 2011-03-10 WO disclosed