SCHEMBL12833452

SCHEMBL12833452

O=C(C[C@H](O)c1ccc(Cl)nc1)N1C(=O)OC[C@@H]1Cc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 12/20 0.38
NAAA Q02083 1/20 0.36
IL6ST P40189 1/20 0.35
FAAH O00519 1/20 0.35
PPARA Q07869 1/20 0.34
CSNK2B P67870 1/20 0.34
CSNK2A1 P68400 1/20 0.34
MAPT P10636 1/20 0.34
KDM1A O60341 1/20 0.34
NAMPT P43490 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL46343 0.85 IDH1 (0.44) IDH1NAAAIL6STFAAHPPARA
SCHEMBL3747623 0.80 CACNA2D1 (0.45) IDH1NAAAPPARA
SCHEMBL3747620 0.80 CACNA2D1 (0.45) IDH1NAAAPPARA
SCHEMBL13654970 0.80 PPARA (0.37) IDH1NAAAIL6STPPARACSNK2B
SCHEMBL9962996 0.78 AGTR2 (0.35) IDH1IL6STFAAHPPARACSNK2B
SCHEMBL1049822 0.76 NAAA (0.46) IDH1NAAAIL6STFAAHPPARA
SCHEMBL2029159 0.76 NAAA (0.46) IDH1NAAAIL6STFAAHPPARA
SCHEMBL1049820 0.76 NAAA (0.46) IDH1NAAAIL6STFAAHPPARA
SCHEMBL17241988 0.76 IDH1 (0.45) IDH1NAAAIL6STFAAHPPARA
SCHEMBL17241987 0.76 IDH1 (0.45) IDH1NAAAIL6STFAAHPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011025774-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME CORP. (US) 2011-03-03 WO disclosed