SCHEMBL12835945

SCHEMBL12835945

CN1CCCC(S(=O)(=O)c2ccc(Br)cc2)C1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.40
LMNA P02545 1/20 0.40
SIGMAR1 Q99720 4/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
HCRTR1 O43613 1/20 0.38
HCRTR2 O43614 1/20 0.38
MMP1 P03956 1/20 0.37
MMP8 P22894 1/20 0.37
MMP13 P45452 1/20 0.37
HRH3 Q9Y5N1 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20284412 0.84 HTR2A (0.49) ATMHTTPOLB
SCHEMBL28897684 0.84 LMNA (0.42) LMNASIGMAR1MAPK1HTTMMP1
SCHEMBL9963142 0.81 HTR6 (0.39) ATMLMNAMAPK1HTTHCRTR1
SCHEMBL14941033 0.81 ATM (0.38) ATMSIGMAR1MAPK1HTTHCRTR1
SCHEMBL5438989 0.81 LMNA (0.47) LMNA
SCHEMBL28022948 0.78 POLB (0.43) POLB
SCHEMBL1939864 0.78 MAPK1 (0.53) MAPK1HTTMMP1MMP8MMP13
SCHEMBL25296150 0.77 MAPK1 (0.56) MAPK1HTTMMP1MMP8MMP13
SCHEMBL14986328 0.76 HTR2A (0.51) HTTPOLB
SCHEMBL14927923 0.76 CA1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8841449-B2 Compounds useful as inhibitors of ATR kinase VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-09-23 US disclosed
US-20130115310-A1 Compounds Useful as Inhibitors of ATR Kinase VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-05-09 US disclosed
WO-2011025690-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME CORP. (US) 2011-03-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130115310-A1 Compounds Useful as Inhibitors of ATR Kinase ATR, CHEK1, CHEK2 ATM 31/4885LMNA 1721/4885SIGMAR1 4783/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.