SCHEMBL12855286

SCHEMBL12855286

CC(C)NC(=O)c1cccc(C(=O)NCc2ccc(-c3ccc(F)c(I)c3)nc2)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 3/20 0.40
MAPK8 P45983 1/20 0.40
MAPK9 P45984 1/20 0.40
ROCK2 O75116 2/20 0.39
ROCK1 Q13464 2/20 0.39
MMP13 P45452 1/20 0.39
ERN1 O75460 1/20 0.38
CTSA P10619 2/20 0.38
POLB P06746 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HTR2C P28335 2/20 0.38
MCHR1 Q99705 2/20 0.38
CNR1 P21554 2/20 0.37
PRKD1 Q15139 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
AVPR1B P47901 1/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8206189 0.89 CNR2 (0.52) CNR2MAPK8MAPK9CTSACNR1
SCHEMBL8199927 0.87 CNR2 (0.50) CNR2POLBSMN1; SMN2CNR1
SCHEMBL8209069 0.85 CNR2 (0.47) CNR2CTSACNR1AVPR1B
SCHEMBL8205711 0.84 SMN1; SMN2 (0.44) MAPK8MAPK9CTSASMN1; SMN2CNR1
SCHEMBL8206930 0.84 MMP13 (0.46) MAPK8MAPK9ROCK2ROCK1MMP13
SCHEMBL8212427 0.84 SMN1; SMN2 (0.41) CNR2MAPK8MAPK9ROCK2ROCK1
SCHEMBL8198357 0.83 CNR1 (0.52) MAPK8MAPK9ROCK1CTSAPOLB
SCHEMBL8198360 0.83 ECE1 (0.46) MAPK8MAPK9ROCK2ROCK1ERN1
SCHEMBL8205692 0.82 MAPK8 (0.47) MAPK8MAPK9ROCK2ROCK1ERN1
SCHEMBL12853352 0.82 CNR2 (0.52) CNR2MMP13CTSACNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8278337-B2 Substituted pyridines that are JNK inhibitors MERCK SHARP & DOHME (US) 2012-10-02 US disclosed