SCHEMBL8205692

SCHEMBL8205692

CC(C)NC(=O)c1cccc(C(=O)NCc2ccc(-c3ccc(N)cc3)nc2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 2/20 0.47
MAPK9 P45984 2/20 0.47
ACVR1 Q04771 1/20 0.44
KLKB1 P03952 2/20 0.42
KLK1 P06870 1/20 0.42
HPGDS O60760 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CNR1 P21554 1/20 0.41
MAPK10 P53779 1/20 0.40
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
HIF1A Q16665 1/20 0.40
SCN9A Q15858 4/20 0.39
HPGD P15428 3/20 0.38
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ERN1 O75460 1/20 0.38
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8198357 0.91 CNR1 (0.52) MAPK8MAPK9HPGDSCNR1ROCK1
SCHEMBL8198360 0.90 ECE1 (0.46) MAPK8MAPK9ACVR1KLKB1KLK1
SCHEMBL8205711 0.90 SMN1; SMN2 (0.44) MAPK8MAPK9HPGDSCNR1HPGD
SCHEMBL8207782 0.88 CA1 (0.49) MAPK8MAPK9KLKB1KLK1CA1
SCHEMBL12853347 0.87 MAPK8 (0.49) MAPK8MAPK9HPGDSMAPK10SCN9A
SCHEMBL12853349 0.87 MAPK8 (0.51) MAPK8MAPK9CA1CA2MAPK10
SCHEMBL8212490 0.85 CA1 (0.46) MAPK8MAPK9KLKB1KLK1CA1
SCHEMBL8206930 0.84 MMP13 (0.46) MAPK8MAPK9HPGDSCNR1ROCK2
SCHEMBL8212427 0.84 SMN1; SMN2 (0.41) MAPK8MAPK9HPGDSCNR1ROCK2
SCHEMBL8209069 0.84 CNR2 (0.47) CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008082487-A2 NOVEL JNK INHIBITORS SCHERING CORPORATION (US) 2008-07-10 WO disclosed