SCHEMBL8198360

SCHEMBL8198360

CC(C)NC(=O)c1cccc(C(=O)NCc2ccc(-c3cccc(N)c3)nc2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 1/20 0.46
MAPK8 P45983 2/20 0.43
MAPK9 P45984 2/20 0.43
MAPK10 P53779 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
HPGDS O60760 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
PRKD1 Q15139 1/20 0.39
ERN1 O75460 1/20 0.39
KLKB1 P03952 1/20 0.39
KLK1 P06870 1/20 0.39
ADORA2A P29274 3/20 0.38
ADORA1 P30542 3/20 0.38
FLT3 P36888 1/20 0.38
TYRO3 Q06418 1/20 0.38
MERTK Q12866 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8205692 0.90 MAPK8 (0.47) MAPK8MAPK9MAPK10HPGDSCA1
SCHEMBL8206930 0.89 MMP13 (0.46) MAPK8MAPK9HPGDSROCK2ROCK1
SCHEMBL8199927 0.88 CNR2 (0.50) CYP11B1HPGDSKLKB1KLK1ADORA2A
SCHEMBL8209069 0.88 CNR2 (0.47) ADORA2AADORA1
SCHEMBL8207800 0.86 ROCK2 (0.47) MAPK8MAPK9MAPK10CA1CA2
SCHEMBL12853352 0.85 CNR2 (0.52)
SCHEMBL12853345 0.85 CTSA (0.47) MAPK8MAPK9MAPK10CYP11B1ADORA2A
SCHEMBL8205721 0.85 MAPK8 (0.47) MAPK8MAPK9MAPK10CA1CA2
SCHEMBL8211821 0.85 ROCK2 (0.47) MAPK8MAPK9MAPK10CA1CA2
SCHEMBL8212427 0.85 SMN1; SMN2 (0.41) MAPK8MAPK9HPGDSROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008082487-A2 NOVEL JNK INHIBITORS SCHERING CORPORATION (US) 2008-07-10 WO disclosed