SCHEMBL12857014

SCHEMBL12857014

N=C(Nc1ccc2ccn(CCCCN)c2c1)c1cccs1

nearest known ligand 0.48

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 19/20 0.48
NOS3 P29474 18/20 0.48
NOS2 P35228 4/20 0.47
ITK Q08881 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15499701 0.90 NOS1 (0.47) NOS1NOS3NOS2
SCHEMBL1122396 0.86 NOS3 (0.62) NOS1NOS3NOS2
SCHEMBL12253664 0.86 NOS1 (0.63) NOS1NOS3NOS2
SCHEMBL12253663 0.85 NOS3 (0.62) NOS1NOS3NOS2
Hydrochloric Acid SCHEMBL1122320 0.85 NOS3 (0.63) NOS1NOS3NOS2
SCHEMBL1122409 0.85 NOS3 (0.65) NOS1NOS3NOS2
SCHEMBL12253662 0.84 NOS3 (0.62) NOS1NOS3NOS2
Hydrochloric Acid SCHEMBL1122252 0.84 NOS3 (0.62) NOS1NOS3NOS2
SCHEMBL12253661 0.83 NOS3 (0.63) NOS1NOS3NOS2
Hydrochloric Acid SCHEMBL1121949 0.83 NOS3 (0.63) NOS1NOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1883451-B9 SUBSTITUTED INDOLE COMPOUNDS HAVING NOS INHIBITORY ACTIVITY NEURAXON INC (CA) 2011-02-09 EP disclosed
EP-1883451-B1 SUBSTITUTED INDOLE COMPOUNDS HAVING NOS INHIBITORY ACTIVITY NEURAXON INC (CA) 2010-11-24 EP disclosed
WO-2010132072-A1 TREATMENT OR PREVENTION OF MIGRAINE BY DOSING AT AURA NEURAXON, INC (CA) 2010-11-18 WO disclosed