SCHEMBL1287902

SCHEMBL1287902

CC(C)c1cn(COCc2ccc(F)cc2)c(=O)[nH]c1=O

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
TK1 P04183 1/20 0.39
MET P08581 1/20 0.38
DAO P14920 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
UPP1 Q16831 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
THRB P10828 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1287942 0.87 ALDH1A1 (0.52) ALDH1A1TK1DAOUPP1MAPK1
SCHEMBL1287949 0.78 HTT (0.36) UPP1KDM4EMAPK1
SCHEMBL7540000 0.76 TK1 (0.46) ALDH1A1TK1DAOUPP1MAPT
SCHEMBL20870268 0.74 GRIA1 (0.38) ALDH1A1CYP2C9KDM4EMAPTMAPK1
SCHEMBL9016400 0.74 UPP1 (0.53) UPP1
SCHEMBL13384426 0.74 UPP1 (0.39) CYP2C9UPP1MAPT
SCHEMBL1287911 0.73 ALDH1A1 (0.44) ALDH1A1DAOL3MBTL1CYP2C9CYP2C19
SCHEMBL6719842 0.71 ALDH1A1 (0.52) ALDH1A1TK1DAOCYP2C9CYP2C19
SCHEMBL13384443 0.71 SMN1; SMN2 (0.40) CYP2C9CYP2C19KDM4EMAPTMAPK1
SCHEMBL13384415 0.70 HPGD (0.66) TK1DAOMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047993-A2 N-HYDROXYPYRIMIDINE-2,4-DIONES AS INHIBITORS OF HIV AND HCV REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2012-04-12 WO disclosed