SCHEMBL1289375

SCHEMBL1289375

CC(C)(N)CCNc1nc(-c2cnc3ccccc3c2)nc2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.54
PDE5A O76074 4/20 0.54
ACP1 P24666 2/20 0.52
MAPK1 P28482 2/20 0.50
MAPT P10636 2/20 0.49
GBA1 P04062 2/20 0.49
RECQL P46063 2/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
TLR9 Q9NR96 1/20 0.49
SLC6A3 Q01959 2/20 0.48
ALDH1A1 P00352 2/20 0.48
KDM4E B2RXH2 2/20 0.47
ROCK2 O75116 1/20 0.47
ROCK1 Q13464 1/20 0.47
PKN2 Q16513 1/20 0.47
LMNA P02545 1/20 0.47
TP53 P04637 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4505205 0.99 KDM1A (0.53) KDM1APDE5AACP1MAPK1MAPT
Hydrochloric Acid SCHEMBL4518504 0.85 PDE5A (0.52) PDE5AACP1MAPK1MAPTGBA1
SCHEMBL10065463 0.80 MAPK1 (0.77) KDM1APDE5AACP1MAPK1MAPT
SCHEMBL23723245 0.80 PDE5A (0.53) PDE5AACP1MAPK1MAPTGBA1
Hydrochloric Acid SCHEMBL4502640 0.79 MAPK1 (0.79) KDM1APDE5AACP1MAPK1GBA1
SCHEMBL17770552 0.76 ROCK2 (0.64) PDE5AACP1MAPK1MAPTGBA1
Hydrochloric Acid SCHEMBL4508477 0.75 PDE5A (0.43) PDE5AACP1MAPK1MAPTGBA1
SCHEMBL20573807 0.74 LATS1 (0.78) ROCK2ROCK1PKN2
SCHEMBL4493556 0.74 CYP1A2 (0.43) PDE5AACP1MAPK1MAPTGBA1
Hydrochloric Acid SCHEMBL4494721 0.73 CYP1A2 (0.43) PDE5AACP1MAPK1MAPTGBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012046207-A1 ANTI-PARASITIC SUBSTITUTED RING FUSED AZINE COMPOUNDS PARACO TECHNOLOGY LIMITED (NZ) 2012-04-12 WO disclosed