SCHEMBL1290780

SCHEMBL1290780

O=C(O)Nc1ccc2c(c1)NC1=C(CN2)C(=O)CC=C1

nearest known ligand 0.31

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.31
ITGA2B P08514 2/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
MEN1 O00255 2/20 0.30
KMT2A Q03164 2/20 0.30
SMYD3 Q9H7B4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1290859 0.82 SMYD3 (0.38) ALDH1A1MAPTMEN1KMT2ASMYD3
SCHEMBL1290611 0.80 SMYD3 (0.38) MEN1KMT2ASMYD3
SCHEMBL7982185 0.77 MEN1 (0.48) ALDH1A1MAPTMEN1KMT2A
SCHEMBL1290996 0.68 HDAC2 (0.48) MAPTMEN1KMT2A
SCHEMBL578342 0.62 SMYD3 (0.61) SMYD3
SCHEMBL29642948 0.62 SMYD3 (0.61) SMYD3
SCHEMBL30950742 0.61 RAB9A (0.37) ALDH1A1MAPTMEN1KMT2A
SCHEMBL2295986 0.61 RAB9A (0.37) ALDH1A1MAPTMEN1KMT2A
SCHEMBL28552531 0.60 AHR (0.50) MAPTMEN1KMT2A
SCHEMBL3060475 0.60 ACVRL1 (0.34) ALDH1A1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012045194-A1 BENZODIAZEPINONES AS FAK INHIBITORS FOR TREATMENT OF CANCER ABBOTT LABORATORIES (US) 2012-04-12 WO disclosed