SCHEMBL13004635

SCHEMBL13004635

Cc1cccc(-c2ccc(-c3ncc(C(=O)O)s3)cc2C#N)c1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 2/20 0.45
HSD17B2 P37059 2/20 0.45
XDH P47989 6/20 0.44
NPC1 O15118 4/20 0.43
RAB9A P51151 4/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
POLB P06746 2/20 0.43
S1PR1 P21453 1/20 0.41
S1PR5 Q9H228 1/20 0.41
ALDH1A1 P00352 3/20 0.40
MAPT P10636 3/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
LRRK2 Q5S007 1/20 0.39
AR P10275 1/20 0.39
GRM5 P41594 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13004936 0.89 XDH (0.45) XDHS1PR1S1PR5
SCHEMBL1331310 0.89 XDH (0.49) XDHNPC1RAB9ASMN1; SMN2POLB
SCHEMBL23794763 0.85 HSD17B1 (0.57) HSD17B1HSD17B2NPC1RAB9ASMN1; SMN2
SCHEMBL13140006 0.81 HDAC3 (0.42) XDHS1PR1S1PR5LRRK2AR
SCHEMBL13004637 0.81 XDH (0.54) XDHSMN1; SMN2S1PR1S1PR5
SCHEMBL13118072 0.81 HSD17B1 (0.46) HSD17B1HSD17B2NPC1RAB9ASMN1; SMN2
SCHEMBL3384040 0.80 XDH (0.60) XDHNPC1RAB9ASMN1; SMN2POLB
SCHEMBL3385772 0.77 XDH (0.46) XDHMAPTGRM5
SCHEMBL23794627 0.76 NPC1 (0.49) XDHNPC1RAB9ASMN1; SMN2POLB
SCHEMBL13004937 0.76 XDH (0.45) HSD17B1HSD17B2XDHARGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1932832-B1 TRIARYLCARBOXYLIC ACID DERIVATIVE ASTELLAS PHARMA INC (JP) 2010-12-01 EP disclosed
EP-1932832-A1 TRIARYLCARBOXYLIC ACID DERIVATIVE Astellas Pharma Inc. (JP) 2008-06-18 EP disclosed