SCHEMBL13005203

SCHEMBL13005203

CC(C)(C)c1ccc2nc(-c3ccccc3)c(CCC(O)CO)cc2c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.36
AKT2 P31751 1/20 0.36
PSMB5 P28074 1/20 0.36
SCN10A Q9Y5Y9 1/20 0.36
PDE10A Q9Y233 1/20 0.35
PTGFR P43088 5/20 0.35
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34
KDM4E B2RXH2 3/20 0.34
ALDH1A1 P00352 3/20 0.34
DHODH Q02127 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
DHFR P00374 1/20 0.32
ACSS2 Q9NR19 1/20 0.32
HPGD P15428 1/20 0.32
MAPK1 P28482 1/20 0.32
CASP1 P29466 1/20 0.32
RAB9A P51151 1/20 0.32
CASP7 P55210 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13005210 0.83 AKT1 (0.39) AKT1AKT2PSMB5SCN10APDE10A
SCHEMBL10102637 0.83 ALDH1A1 (0.37) KDM4EALDH1A1CASP1RAB9ACASP7
SCHEMBL10102675 0.78 PSMB5 (0.43) AKT1AKT2PSMB5PDE10ADHFR
SCHEMBL10102678 0.77 AKT1 (0.37) AKT1AKT2PSMB5PDE10APTGFR
SCHEMBL10107981 0.75 KIF11 (0.38) PTGFRKDM4EALDH1A1HPGD
SCHEMBL13004928 0.74 DHODH (0.46) PTGFRRXRARXRBRXRGKDM4E
SCHEMBL13005241 0.74 GPBAR1 (0.40) KDM4EL3MBTL1
SCHEMBL10102671 0.73 DHODH (0.46) RXRARXRBRXRGKDM4EDHODH
SCHEMBL3386183 0.73 PIK3CG (0.40) SCN10AALDH1A1HPGDRAB9A
SCHEMBL10102677 0.73 VSIR (0.38) AKT1AKT2PSMB5PTGFRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891011-B1 TETRAHYDROQUINOLINES USED IN THE FORM OF MODULATORS OF MITOTIC MOTOR-PROTEINS EG5 MERCK PATENT GMBH (DE) 2010-12-08 EP disclosed