SCHEMBL13005654

SCHEMBL13005654

CC(C)Cc1cccc(CN(CCN(C)C)CC2CC3C=CC2C3)c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CALM1 P0DP23 1/20 0.37
CAMKK2 Q96RR4 1/20 0.37
KDM4E B2RXH2 6/20 0.32
ALDH1A1 P00352 3/20 0.32
TDP1 Q9NUW8 1/20 0.32
MEN1 O00255 3/20 0.31
KMT2A Q03164 3/20 0.31
HTT P42858 1/20 0.31
BCHE P06276 1/20 0.31
TSHR P16473 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C19 P33261 1/20 0.30
ATM Q13315 1/20 0.30
CETP P11597 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13060702 0.88 CALM1 (0.38) CALM1CAMKK2KDM4EALDH1A1TDP1
SCHEMBL13005651 0.80 CALM1 (0.36) CALM1CAMKK2ALDH1A1
SCHEMBL13005691 0.79 OPRM1 (0.43) CALM1CAMKK2
SCHEMBL13005432 0.78 OPRM1 (0.44) CALM1CAMKK2ALDH1A1
SCHEMBL13005625 0.77 BCHE (0.47) CALM1CAMKK2MEN1KMT2ABCHE
SCHEMBL13005440 0.76 CALM1 (0.59) CALM1CAMKK2KDM4EALDH1A1MEN1
SCHEMBL13005422 0.75 CALM1 (0.48) CALM1CAMKK2KDM4EALDH1A1MEN1
SCHEMBL13005722 0.74 CALM1 (0.48) CALM1CAMKK2KDM4EALDH1A1TDP1
SCHEMBL13005681 0.74 CALM1 (0.48) CALM1CAMKK2KDM4EALDH1A1MEN1
SCHEMBL13005558 0.74 KDM4E (0.54) CALM1CAMKK2KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7851637-B2 Compounds and methods for inhibiting the interaction of BCL proteins with binding partners INFINITY PHARMACEUTICALS, INC. (US) 2010-12-14 US disclosed