SCHEMBL13007458

SCHEMBL13007458

O=C(Nc1ccccc1NCCN1CCCC1)NC1CCCc2ccccc21

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 2/20 0.61
TAS1R1 Q7RTX1 2/20 0.61
NPSR1 Q6W5P4 1/20 0.61
ALDH1A1 P00352 2/20 0.59
KDM4E B2RXH2 1/20 0.59
GAA P10253 1/20 0.59
HPGD P15428 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
KMT2A Q03164 6/20 0.58
MEN1 O00255 1/20 0.57
HTT P42858 1/20 0.54
LMNA P02545 2/20 0.53
ATM Q13315 1/20 0.52
EPHX1 P07099 1/20 0.51
EPHX2 P34913 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13007504 0.82 KMT2A (0.68) TAS1R3TAS1R1NPSR1ALDH1A1KDM4E
SCHEMBL701314 0.76 TAS1R3 (1.00) TAS1R3TAS1R1NPSR1ALDH1A1KDM4E
SCHEMBL703637 0.76 TAS1R3 (1.00) TAS1R3TAS1R1NPSR1ALDH1A1KDM4E
SCHEMBL7780152 0.75 HRH3 (0.54) ALDH1A1KDM4E
SCHEMBL30046159 0.73 HTT (0.68) TAS1R3TAS1R1NPSR1ALDH1A1HPGD
SCHEMBL30751972 0.73 HTT (0.68) TAS1R3TAS1R1NPSR1ALDH1A1HPGD
SCHEMBL1441796 0.73 HTT (0.68) TAS1R3TAS1R1NPSR1ALDH1A1HPGD
SCHEMBL2358933 0.73 HTT (0.68) TAS1R3TAS1R1NPSR1ALDH1A1HPGD
SCHEMBL31730298 0.72 TAOK3 (0.64) ALDH1A1HPGD
SCHEMBL5652051 0.72 TAOK3 (0.64) ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1861377-B1 BENZIMIDAZOLONE DERIVATIVES AS CB2 RECEPTOR LIGANDS PFIZER (US) 2010-12-29 EP disclosed
WO-2008032164-A2 BENZIMIDAZOLONE DERIVATIVES PFIZER PRODUCTS INC. (US) 2008-03-20 WO disclosed