SCHEMBL1301622

SCHEMBL1301622

Clc1cccc(C[Zn]Br)c1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PNMT P11086 2/20 0.56
TAAR1 Q96RJ0 3/20 0.52
IDO1 P14902 3/20 0.50
CYP3A4 P08684 2/20 0.50
AGXT P21549 2/20 0.50
HTR3E A5X5Y0 3/20 0.47
HTR3B O95264 3/20 0.47
HTR3A P46098 3/20 0.47
HTR3D Q70Z44 3/20 0.47
HTR3C Q8WXA8 3/20 0.47
CHRM2 P08172 1/20 0.46
SIGMAR1 Q99720 1/20 0.46
AOC3 Q16853 1/20 0.44
MAOB P27338 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3216346 0.81 TAAR1 (0.57) PNMTTAAR1IDO1CYP3A4AGXT
SCHEMBL2256351 0.79 PNMT (0.58) PNMTTAAR1IDO1CYP3A4AGXT
SCHEMBL2216304 0.77 PNMT (0.56) PNMTTAAR1IDO1CYP3A4AGXT
SCHEMBL2436 0.76
SCHEMBL5733314 0.76 PNMT (0.60) PNMTTAAR1IDO1CYP3A4AGXT
SCHEMBL29353832 0.76
Bromide SCHEMBL1301106 0.76 PNMT (0.54) PNMTTAAR1IDO1CYP3A4AGXT
SCHEMBL12050856 0.75 TAAR1 (0.74) PNMTTAAR1IDO1CYP3A4AGXT
SCHEMBL3300276 0.75 PNMT (0.65) PNMTTAAR1IDO1CYP3A4AGXT
SCHEMBL1001013 0.74 PNMT (0.58) PNMTTAAR1IDO1CYP3A4AGXT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137162-B1 ORGANIC COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2018-08-01 EP disclosed
US-8536168-B2 Benzyl and pyridinyl derivatives as modulators of the hedgehog signaling pathway NOVARTIS AG (CH) 2013-09-17 US disclosed
US-20110269741-A1 NOVEL COMPOSITIONS AND METHODS OF USE ARDEA BIOSCIENCES, INC. (US) 2011-11-03 US disclosed
US-20100069368-A1 Organic Compounds and Their Uses NOVARTIS AG (CH) 2010-03-18 US disclosed
EP-2137162-A1 ORGANIC COMPOUNDS AND THEIR USES Novartis Ag (CH) 2009-12-30 EP disclosed
WO-2008110611-A1 ORGANIC COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2008-09-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110269741-A1 NOVEL COMPOSITIONS AND METHODS OF USE TYMP, SAMHD1, PNP PNMT 1050/4885TAAR1 4760/4885IDO1 532/4885
US-20100069368-A1 Organic Compounds and Their Uses SHH, GLI1, VHL PNMT 1194/4885TAAR1 3136/4885IDO1 3858/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.