SCHEMBL13037152

SCHEMBL13037152

CCOC(=O)C(C)(C)c1cc(C)nc(-n2ccnc2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
KMT2A Q03164 3/20 0.42
KDM4E B2RXH2 3/20 0.42
MEN1 O00255 2/20 0.42
MAPT P10636 2/20 0.42
MITF O75030 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NOS2 P35228 3/20 0.42
HPGD P15428 1/20 0.41
CXCR2 P25025 1/20 0.41
TDP1 Q9NUW8 2/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
ATM Q13315 1/20 0.41
LMNA P02545 1/20 0.39
CD38 P28907 5/20 0.39
CYP1A2 P05177 4/20 0.39
CYP2C19 P33261 1/20 0.39
CYP26A1 O43174 1/20 0.38
CNR2 P34972 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3558930 0.84 NOS2 (0.43) ALDH1A1KMT2AKDM4EMEN1NOS2
SCHEMBL3559596 0.83 NOS2 (0.42) ALDH1A1KMT2AKDM4EMEN1NOS2
SCHEMBL3565421 0.81 ALDH1A1 (0.41) ALDH1A1KMT2AKDM4EMEN1MAPT
SCHEMBL3565426 0.81 ALDH1A1 (0.41) ALDH1A1KMT2AKDM4EMEN1MAPT
SCHEMBL25485897 0.78 KDM4E (0.45) ALDH1A1KMT2AKDM4EMEN1MAPT
SCHEMBL3563653 0.77 NOS2 (0.46) ALDH1A1KMT2AKDM4EMEN1NOS2
SCHEMBL13074178 0.77 NOS2 (0.43) NOS2CD38CYP1A2CYP2C19
SCHEMBL3573524 0.75 NOS2 (0.46) ALDH1A1KMT2AKDM4EMEN1MAPT
SCHEMBL3559939 0.75 NOS2 (0.46) ALDH1A1KMT2AKDM4EMEN1NOS2
SCHEMBL3558712 0.75 NOS2 (0.46) ALDH1A1KMT2AKDM4EMEN1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7825256-B2 Inducible nitric oxide synthase dimerization inhibitors KALYPSYS, INC. (US) 2010-11-02 US disclosed