SCHEMBL13074178

SCHEMBL13074178

Cc1cc(C(C)(C)C(=O)C2CO2)nc(-n2ccnc2)n1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 13/20 0.43
CD38 P28907 5/20 0.38
CYP1A2 P05177 4/20 0.38
CYP2C19 P33261 1/20 0.38
NOS1 P29475 3/20 0.37
CHEK1 O14757 1/20 0.35
ATR Q13535 1/20 0.35
PDCD1 Q15116 1/20 0.35
ATRIP Q8WXE1 1/20 0.35
CD274 Q9NZQ7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3558930 0.82 NOS2 (0.43) NOS2CD38CYP1A2CYP2C19
SCHEMBL3559596 0.81 NOS2 (0.42) NOS2CD38CYP1A2CYP2C19
SCHEMBL13037152 0.77 ALDH1A1 (0.42) NOS2CD38CYP1A2CYP2C19
SCHEMBL3573524 0.73 NOS2 (0.46) NOS2CD38CYP1A2CYP2C19
SCHEMBL3563653 0.73 NOS2 (0.46) NOS2CD38CYP1A2CYP2C19NOS1
SCHEMBL3558712 0.73 NOS2 (0.46) NOS2CD38CYP1A2CYP2C19NOS1
SCHEMBL3568833 0.72 NOS2 (0.40) NOS2CD38CYP1A2CYP2C19
SCHEMBL3568834 0.72 NOS2 (0.40) NOS2CD38CYP1A2CYP2C19
SCHEMBL13037188 0.71 LMNA (0.50) NOS2CYP1A2CYP2C19
SCHEMBL3559939 0.70 NOS2 (0.46) NOS2CD38CYP1A2CYP2C19NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7825256-B2 Inducible nitric oxide synthase dimerization inhibitors KALYPSYS, INC. (US) 2010-11-02 US disclosed