SCHEMBL13049580

SCHEMBL13049580

CC[C@@]12c3c4ccc(O)c3OC1C(=O)CCC2C(NCC1CC1)C4

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 8/20 0.49
OPRD1 P41143 8/20 0.49
OPRK1 P41145 7/20 0.49
CYP2D6 P10635 2/20 0.42
CHRNA7 P36544 1/20 0.42
CYP1A2 P05177 1/20 0.42
PKM P14618 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12945210 0.80 OPRD1 (0.39) OPRM1OPRD1OPRK1
SCHEMBL21859260 0.78 OPRD1 (0.55) OPRM1OPRD1OPRK1CYP2D6CHRNA7
SCHEMBL19194810 0.77 OPRM1 (0.51) OPRM1OPRD1OPRK1
SCHEMBL19777068 0.77 OPRD1 (0.37) OPRM1OPRD1OPRK1
SCHEMBL19198659 0.76 OPRM1 (0.34) OPRM1OPRD1OPRK1
SCHEMBL20170829 0.76 OPRD1 (0.46) OPRM1OPRD1OPRK1
SCHEMBL21859469 0.75 OPRM1 (0.51) OPRM1OPRD1OPRK1CYP2D6CHRNA7
SCHEMBL13257561 0.74 OPRM1 (0.54) OPRM1OPRD1OPRK1CYP2D6
SCHEMBL14772785 0.74 OPRM1 (0.54) OPRM1OPRD1OPRK1CYP2D6
SCHEMBL13357084 0.74 OPRM1 (0.54) OPRM1OPRD1OPRK1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010144641-A1 PREPARATION OF 6-ALPHA-AMINO N-SUBSTITUTED MORPHINANS BY CATALYTIC HYDROGEN TRANSFER MALLINCKRODT INC. (US) 2010-12-16 WO disclosed
WO-2010039222-A2 PROCESSES FOR THE SELECTIVE AMINATION OF KETOMORPHINANS MALLINCKRODT INC. (US) 2010-04-08 WO disclosed