SCHEMBL13069607

SCHEMBL13069607

O=CC1CC1(C(=O)O)c1ccc2nccnc2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.39
KDM4E B2RXH2 6/20 0.39
MAPT P10636 6/20 0.39
SMN1; SMN2 Q16637 6/20 0.39
KMT2A Q03164 6/20 0.39
HPGD P15428 6/20 0.35
CASP1 P29466 3/20 0.35
HSD17B10 Q99714 3/20 0.35
MAPK1 P28482 1/20 0.35
TP53 P04637 4/20 0.35
CASP7 P55210 2/20 0.35
NPC1 O15118 9/20 0.33
RAB9A P51151 9/20 0.33
POLB P06746 3/20 0.33
GAA P10253 3/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC8 Q9BY41 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6024290 0.75 CCR2 (0.43) CYP3A4CYP1A2CYP2C9CYP2C19TSHR
SCHEMBL13180805 0.75 PIK3CD (0.35) ALDH1A1KDM4EMAPTSMN1; SMN2KMT2A
SCHEMBL3742183 0.75 CCR2 (0.43) CYP3A4CYP1A2CYP2C9CYP2C19TSHR
SCHEMBL1721474 0.71 AKR1C3 (0.44) ALDH1A1KDM4EMAPTSMN1; SMN2KMT2A
SCHEMBL3094127 0.65 ALDH1A1 (0.45) ALDH1A1KDM4EMAPTSMN1; SMN2KMT2A
SCHEMBL3753394 0.62 CCR2 (0.41) HDAC3HDAC1CYP3A4CYP1A2CYP2C9
SCHEMBL3753398 0.62 CCR2 (0.41) HDAC3HDAC1CYP3A4CYP1A2CYP2C9
SCHEMBL3753400 0.62 CCR2 (0.41) HDAC3HDAC1CYP3A4CYP1A2CYP2C9
SCHEMBL3094130 0.61 MAPT (0.36) ALDH1A1KDM4EMAPTSMN1; SMN2KMT2A
SCHEMBL13736220 0.61 RAB9A (0.35) ALDH1A1KDM4ESMN1; SMN2KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919908-B1 TRIAZOLE DERIVATIVES AS MODULATORS OF DOPAMINE D3 RECEPTORS GLAXO GROUP LTD (GB) 2010-11-10 EP disclosed