SCHEMBL13070513

SCHEMBL13070513

CCc1c2[n+](c(Cl)c3c(OC)c(OC)ccc13)CCc1cc(O)c(O)cc1-2

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 13/20 0.48
RAC1 P63000 2/20 0.45
CYP1B1 Q16678 1/20 0.45
ACHE P22303 1/20 0.45
MAOB P27338 1/20 0.45
KDM1A O60341 3/20 0.40
CYP3A4 P08684 2/20 0.40
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
RAD52 P43351 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TRPC5 Q9UL62 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13070786 0.88 COL1A1 (0.45) P2RX7RAC1CYP1B1ACHEMAOB
SCHEMBL13070792 0.87 KDM1A (0.49) P2RX7RAC1CYP1B1ACHEMAOB
SCHEMBL298694 0.86 P2RX7 (0.66) P2RX7CYP1B1ACHEKDM1ACYP3A4
SCHEMBL13070373 0.78 P2RX7 (0.74) P2RX7RAC1CYP1B1ACHEMAOB
SCHEMBL298485 0.76 P2RX7 (0.55) P2RX7CYP1B1ACHEKDM1ACYP3A4
SCHEMBL13070312 0.76 RAC1 (0.60) RAC1CYP1B1ACHEMAOBKDM1A
SCHEMBL298971 0.74 P2RX7 (0.55) P2RX7CYP1B1ACHEKDM1ACYP3A4
SCHEMBL13070517 0.70 BCHE (0.44) P2RX7RAC1CYP1B1ACHEMAOB
SCHEMBL14513596 0.68 P2RX7 (0.84) P2RX7KDM1A
SCHEMBL13071078 0.68 KDM1A (0.81) P2RX7RAC1CYP1B1ACHEMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010128061-A1 NOVEL ISOQUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2010-11-11 WO disclosed