SCHEMBL13071422

SCHEMBL13071422

CC1(S(=O)(=O)NC(=O)[C@H]2C[C@H]2/C=C\CCCCC[C@H](Nc2ccccn2)C(=O)N2CCC[C@H]2C(N)=O)CC1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
F2 P00734 2/20 0.34
F10 P00742 1/20 0.34
ACE P12821 1/20 0.33
PRSS1 P07477 1/20 0.33
PRSS2 P07478 1/20 0.33
PRSS3 P35030 1/20 0.33
TRHR P34981 1/20 0.33
OPRM1 P35372 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12831720 0.90 ACE (0.37) F2ACEPRSS1PRSS2PRSS3
SCHEMBL13071413 0.88 TRHR (0.32) TRHR
SCHEMBL13071426 0.88 HTT (0.37) TRHR
SCHEMBL13071914 0.87 F2 (0.33) F2ACEPRSS1PRSS2PRSS3
SCHEMBL13071629 0.86 ALDH1A1 (0.36) F2ACEPRSS1PRSS2PRSS3
SCHEMBL13071627 0.86 ELANE (0.34)
SCHEMBL13071403 0.85 USP2 (0.34) F2ACEPRSS1PRSS2PRSS3
SCHEMBL12831783 0.85 F2R (0.34) F2ACEPRSS1PRSS2PRSS3
SCHEMBL13072075 0.85 XIAP (0.31) F2F10TRHROPRM1
SCHEMBL13071626 0.84 DPP4 (0.36) F2ACEPRSS1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009142842-A9 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2010-11-25 WO disclosed
WO-2009142842-A2 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2009-11-26 WO disclosed