SCHEMBL13072089

SCHEMBL13072089

NC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCCC/C=C\[C@@H]1C[C@@H]1C(=O)NS(=O)(=O)C1CC1)Nc1cc(F)c(Cl)c(Cl)c1

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
F2R P25116 2/20 0.33
ACE P12821 1/20 0.31
DPP4 P27487 1/20 0.31
DPP8 Q6V1X1 1/20 0.31
DPP9 Q86TI2 1/20 0.31
DPP7 Q9UHL4 1/20 0.31
TRHR P34981 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13072090 0.90 HTT (0.38) ACETRHR
SCHEMBL13071524 0.88 HTR1A (0.36) ACEDPP4TRHR
SCHEMBL13071668 0.88 ACE (0.33) ACETRHR
SCHEMBL13072094 0.87 USP2 (0.34) F2RACE
SCHEMBL13071393 0.86 DPP4 (0.32) F2RDPP4TRHR
SCHEMBL13071425 0.86 ACE (0.38) ACEDPP4TRHR
SCHEMBL13071878 0.86 XIAP (0.34) F2RACEDPP4
SCHEMBL13071521 0.82 CFD (0.39)
SCHEMBL12831783 0.80 F2R (0.34) F2RACE
SCHEMBL13072075 0.80 XIAP (0.31) TRHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009142842-A9 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2010-11-25 WO disclosed
WO-2009142842-A2 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2009-11-26 WO disclosed