SCHEMBL1307379

SCHEMBL1307379

COCCCOc1ccnc(CS(=O)(=O)c2nc3ccccc3[nH]2)c1C

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.63
CYP2C9 P11712 5/20 0.63
WDR5 P61964 4/20 0.63
ALDH1A1 P00352 4/20 0.63
LMNA P02545 4/20 0.63
ENGASE Q8NFI3 3/20 0.63
MAPT P10636 3/20 0.63
DDAH1 O94760 2/20 0.63
ADORA3 P0DMS8 2/20 0.63
HPGD P15428 2/20 0.63
TBXA2R P21731 2/20 0.63
NPY1R P25929 2/20 0.63
ADORA1 P30542 2/20 0.63
OPRM1 P35372 2/20 0.63
HTR3A P46098 2/20 0.63
FASN P49327 2/20 0.63
SARM1 Q6SZW1 2/20 0.63
ABCG2 Q9UNQ0 2/20 0.63
HTR1A P08908 1/20 0.63
IDE P14735 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30905609 1.00 KMT2A (0.63) KMT2ACYP2C9WDR5ALDH1A1LMNA
SCHEMBL6600439 0.99 CYP2C9 (0.62) KMT2ACYP2C9WDR5ALDH1A1LMNA
SCHEMBL6600434 0.99 KMT2A (0.62) KMT2ACYP2C9WDR5ALDH1A1LMNA
SCHEMBL10121508 0.89 KMT2A (0.62) KMT2ACYP2C9WDR5ALDH1A1LMNA
SCHEMBL23988420 0.88 CYP2C9 (0.51) KMT2ACYP2C9WDR5ALDH1A1LMNA
SCHEMBL23988519 0.86 CYP2C9 (0.53) KMT2ACYP2C9WDR5ALDH1A1LMNA
SCHEMBL5414007 0.85 KMT2A (0.60) KMT2ACYP2C9WDR5ALDH1A1LMNA
SCHEMBL23988509 0.84 CYP2C9 (0.47) KMT2ACYP2C9WDR5ALDH1A1LMNA
SCHEMBL2851048 0.84 KMT2A (0.59) KMT2ACYP2C9WDR5ALDH1A1LMNA
SCHEMBL2851052 0.84 KMT2A (0.59) KMT2ACYP2C9WDR5ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 42 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111714639-A Composition comprising histamine release-promoting substance and benzimidazole derivative 黄泳华 2020-09-29 CN claimed
CN-111084886-A Composition comprising fatty acid or derivative thereof and benzimidazole derivative 黄泳华 2020-05-01 CN claimed
CN-118010878-A Determination method and application of impurities in sodium rabeprazole enteric-coated preparation 丽珠集团丽珠制药厂 2024-05-10 CN disclosed
CN-118010878-A Determination method and application of impurities in sodium rabeprazole enteric-coated preparation 丽珠集团丽珠制药厂 2024-05-10 CN disclosed
US-20220202796-A1 CXCL10 Inhibitors LAPKO INC, dba AFECTA PHARMACEUTICALS 2022-06-30 US disclosed
US-20210338650-A1 CXCL10 Inhibitors AFECTA PHARMACEUTICALS, INC. (US) 2021-11-04 US disclosed
CN-111714639-A Composition comprising histamine release-promoting substance and benzimidazole derivative 黄泳华 2020-09-29 CN disclosed
CN-111084886-A Composition comprising fatty acid or derivative thereof and benzimidazole derivative 黄泳华 2020-05-01 CN disclosed
CN-103483320-B Synthetic method of Rabeprazole Sulfone (2-[[[4-(3-methoxy propoxy)-3-methyl-2-pyridyl] methyl] sulfonyl]-1H-benzimidazole) JILIN XIUZHENG PHARMACEUTICAL NEW MEDICINE DEV CO LTD 2014-12-03 CN disclosed
CN-103483320-B Synthetic method of Rabeprazole Sulfone (2-[[[4-(3-methoxy propoxy)-3-methyl-2-pyridyl] methyl] sulfonyl]-1H-benzimidazole) JILIN XIUZHENG PHARMACEUTICAL NEW MEDICINE DEV CO LTD 2014-12-03 CN disclosed
CN-103483320-A Synthetic method of Rabeprazole Sulfone (2-[[[4-(3-methoxy propoxy)-3-methyl-2-pyridyl] methyl] sulfonyl]-1H-benzimidazole) JILIN XIUZHENG PHARMACEUTICAL NEW MEDICINE DEV CO LTD 2014-01-01 CN disclosed
EP-1775292-A1 SALTS OF BENZIMIDAZOLE DERIVATIVE WITH AMINES AND PROCESS FOR PRODUCTION THEREOF Eisai R&D Management Co., Ltd. (JP) 2007-04-18 EP disclosed
WO-2007023393-A2 NOVEL PROCESSES FOR THE PRODUCTION OF AMORPHOUS RABEPRAZOLE SODIUM MEDICHEM, S.A. (US) 2007-03-01 WO disclosed
WO-2007023393-A2 NOVEL PROCESSES FOR THE PRODUCTION OF AMORPHOUS RABEPRAZOLE SODIUM MEDICHEM, S.A. (US) 2007-03-01 WO disclosed
WO-2007023393-A2 NOVEL PROCESSES FOR THE PRODUCTION OF AMORPHOUS RABEPRAZOLE SODIUM MEDICHEM, S.A. (US) 2007-03-01 WO disclosed
EP-1409478-B1 IMPROVED PROCESS FOR PREPARING BENZIMIDAZOLE-TYPE COMPOUNDS JANSSEN PHARMACEUTICA NV (BE) 2006-03-29 EP disclosed
US-6919459-B2 Process for preparing benzimidazole-type compounds JANSSEN PHARMACEUTICA N.V. (BE) 2005-07-19 US disclosed
US-20040209918-A1 Process for preparing benzimidazole-type compounds JANSSEN PHARMACEUTICA N.V. (BE) 2004-10-21 US disclosed
EP-1409478-A1 IMPROVED PROCESS FOR PREPARING BENZIMIDAZOLE-TYPE COMPOUNDS JANSSEN PHARMACEUTICA N.V. (BE) 2004-04-21 EP disclosed
WO-2003008406-A1 IMPROVED PROCESS FOR PREPARING BENZIMIDAZOLE-TYPE COMPOUNDS JANSSEN PHARMACEUTICA N.V. (BE) 2003-01-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040209918-A1 Process for preparing benzimidazole-type compounds SQOR, CYP2B6, CYP3A5 KMT2A 3547/4885CYP2C9 27/4885WDR5 4069/4885
US-20220202796-A1 CXCL10 Inhibitors CXCL10, CCL5, CCL11 KMT2A 3380/4885CYP2C9 4152/4885WDR5 3395/4885
US-20210338650-A1 CXCL10 Inhibitors CXCL10, CCL5, CCL11 KMT2A 3380/4885CYP2C9 4152/4885WDR5 3395/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.