SCHEMBL130757

SCHEMBL130757

Cn1ccc2c(Cl)ncnc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.46
SLC22A12 Q96S37 1/20 0.44
ABL1 P00519 1/20 0.42
BCR P11274 1/20 0.42
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
FGFR1 P11362 2/20 0.38
FGFR4 P22455 2/20 0.38
RAF1 P04049 1/20 0.36
BRAF P15056 1/20 0.36
KDR P35968 1/20 0.36
MEN1 O00255 1/20 0.34
NR2F2 P24468 1/20 0.34
KMT2A Q03164 1/20 0.34
TP53 P04637 1/20 0.34
CHRNA7 P36544 1/20 0.34
HTR3A P46098 1/20 0.34
PRMT5 O14744 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29407694 1.00 NOTUM (0.46) NOTUMSLC22A12ABL1BCRPDE4A
SCHEMBL256213 0.78 NOTUM (0.47) NOTUMABL1BCRTP53CHRNA7
SCHEMBL4086353 0.77 SLC22A12 (0.42) SLC22A12PDE4APDE4BPDE4CPDE4D
SCHEMBL21822975 0.77 ADORA2A (0.41) NOTUMSLC22A12ABL1BCRPDE4A
SCHEMBL23104228 0.76 NOTUM (0.46) NOTUMABL1BCRRAF1BRAF
SCHEMBL10051003 0.76 PI4KA (0.52) NOTUMABL1BCRMEN1KMT2A
SCHEMBL125104 0.76 NOTUM (0.46) NOTUMABL1BCRRAF1BRAF
SCHEMBL22508902 0.76 SLC22A12 (0.44) SLC22A12PDE4APDE4BPDE4CPDE4D
SCHEMBL19465328 0.76 SLC22A12 (0.44) SLC22A12PDE4APDE4BPDE4CPDE4D
SCHEMBL18572036 0.76 SLC22A12 (0.48) NOTUMSLC22A12PDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 230 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4306529-B1 FGFR INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS INC (US) 2026-01-21 EP disclosed
US-12522605-B2 FGFR inhibitors and methods of use thereof RELAY THERAPEUTICS, INC. (US) 2026-01-13 US disclosed
US-12390463-B2 Dosage forms and regimens for amino acid compounds PLIANT THERAPEUTICS, INC. (US) 2025-08-19 US disclosed
US-20250223288-A1 AMINO ACID COMPOUNDS AND METHODS OF USE PLIANT THERAPEUTICS, INC. 2025-07-10 US disclosed
WO-2025083426-A1 NEW TREATMENTS FOR PAIN SEVENLESS THERAPEUTICS LIMITED (GB) 2025-04-24 WO disclosed
EP-4520329-A2 TREATMENT OF RESPIRATORY DISEASES WITH AMINO ACID COMPOUNDS Pliant Therapeutics, Inc. (US) 2025-03-12 EP disclosed
EP-4509512-A2 AMINO ACID COMPOUNDS AND METHODS OF USE Pliant Therapeutics, Inc. (US) 2025-02-19 EP disclosed
EP-4499616-A1 SPIROBICYCLIC COMPOUNDS Acerand Therapeutics (Hong Kong) Limited (HK) 2025-02-05 EP disclosed
US-11999758-B2 Inhibitors of the YAP/TAZ-TEAD interaction and their use in the treatment of cancer INVENTIVA (FR) 2024-06-04 US disclosed
WO-2024091370-A1 5,6-FUSED BICYCLIC HETEROAROMATIC COMPOUNDS ACERAND THERAPEUTICS (USA) LIMITED (US) 2024-05-02 WO disclosed
CN-1524080-A Phthalatyinone-piperidino-derivatives as pde4 inhibitors ��̹��ҽҩ��˾ 2004-08-25 CN disclosed
WO-2004056830-A1 PYRROLOPYRIMIDINE DERIVATIVES PFIZER PRODUCTS INC. (US) 2004-07-08 WO disclosed
US-20040067946-A1 Phthalatyinone-piperidino-derivatives as pde4 inhibitors TAKEDA GMBH (DE) 2004-04-08 US disclosed
US-20040053924-A1 4-Substituted 7-aza-indolin-2-ones and their use as protein kinase inhibitors SUGEN, INC. 2004-03-18 US disclosed
WO-2004007479-A1 3-GUANIDINOCARBONYL-1-HETEROARYL-INDOLE DERIVATIVES, PREPARATION PROCESS, THEIR USE AS MEDICAMENTS, AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2004-01-22 WO disclosed
EP-1362044-A1 PHTHALAZINONE-PIPERIDINO-DERIVATIVES AS PDE4 INHIBITORS ALTANA Pharma AG (DE) 2003-11-19 EP disclosed
US-6610688-B2 For therapy of blood vessel proliferative disorders; fibrotic disorders; mesangial cell proliferative disorders; metabolic disorders; allergies; asthma; thrombosis; nervous system diseases; and cancer SUGEN, INC. 2003-08-26 US disclosed
US-20020183319-A1 4-substituted 7-aza-indolin-2-ones and their use as protein kinase inhibitors SUGEN, INC. 2002-12-05 US disclosed
WO-2002064584-A1 PHTHALAYINONE-PIPERIDINO-DERIVATIVES AS PDE4 INHIBITORS ALTANA PHARMA AG (DE) 2002-08-22 WO disclosed
WO-1993018035-A1 ANGIOTENSIN II RECEPTOR ANTAGONISTS ABBOTT LABORATORIES (US) 1993-09-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040053924-A1 4-Substituted 7-aza-indolin-2-ones and their use as protein kinase inhibitors CDKN1A, CSNK1A1, CDK2 NOTUM 4602/4885SLC22A12 3572/4885ABL1 33/4885
US-20020183319-A1 4-substituted 7-aza-indolin-2-ones and their use as protein kinase inhibitors CDKN1A, CDK7, CDK2 NOTUM 4582/4885SLC22A12 3013/4885ABL1 30/4885
US-20040067946-A1 Phthalatyinone-piperidino-derivatives as pde4 inhibitors PDE4A, PDE4B, PDE5A NOTUM 2311/4885SLC22A12 1649/4885ABL1 1992/4885
US-12390463-B2 Dosage forms and regimens for amino acid compounds ITGB6, ITGA6, ITGAV NOTUM 4360/4885SLC22A12 326/4885ABL1 955/4885
US-11999758-B2 Inhibitors of the YAP/TAZ-TEAD interaction and their use in the treatment of cancer YAP1, TEAD2, YES1 NOTUM 4397/4885SLC22A12 3540/4885ABL1 31/4885
US-20250223288-A1 AMINO ACID COMPOUNDS AND METHODS OF USE ITGB6, ITGA6, ITGA5 NOTUM 3976/4885SLC22A12 468/4885ABL1 697/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.