SCHEMBL13076397

SCHEMBL13076397

CCCNc1ccc(N(C)C(=O)OC(C)(C)C)cc1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 5/20 0.41
PTGER4 P35408 4/20 0.39
GAA P10253 3/20 0.37
ALDH1A1 P00352 3/20 0.37
MAPT P10636 3/20 0.37
KDM4E B2RXH2 2/20 0.37
THRB P10828 1/20 0.37
HPGD P15428 1/20 0.37
HTT P42858 1/20 0.37
GFER P55789 1/20 0.37
PLEC Q15149 1/20 0.37
BRD4 O60885 1/20 0.36
PAX8 Q06710 1/20 0.36
HSD17B10 Q99714 1/20 0.36
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
NCOR2 Q9Y618 1/20 0.35
ALOX15 P16050 1/20 0.34
PRSS1 P07477 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13076214 0.81 HCAR3 (0.54) PTGER4ALDH1A1MAPTKDM4ENPC1
SCHEMBL397497 0.80 BRD4 (0.41) AAK1GAAALDH1A1MAPTKDM4E
SCHEMBL398694 0.79 BRD4 (0.38) AAK1MAPTKDM4EBRD4PAX8
SCHEMBL13076223 0.77 PTGER4 (0.56) PTGER4GAAALDH1A1MAPTKDM4E
SCHEMBL15156279 0.76 BRD4 (0.42) AAK1ALDH1A1MAPTBRD4PAX8
SCHEMBL13076791 0.75 CA12 (0.42) AAK1PTGER4GAAALDH1A1MAPT
SCHEMBL15156318 0.74 ALDH1A1 (0.46) AAK1GAAALDH1A1MAPTKDM4E
SCHEMBL30369986 0.73 S100B (0.42) AAK1ALDH1A1THRBBRD4PAX8
SCHEMBL18157854 0.73 S100B (0.42) AAK1ALDH1A1THRBBRD4PAX8
SCHEMBL397342 0.73 BRD4 (0.40) AAK1GAAKDM4EHTTBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010126922-A1 BENZIMIDAZOLECARBOXAMIDES AS INHIBITORS OF FAK GLAXOSMITHKLINE LLC (US) 2010-11-04 WO disclosed