SCHEMBL13077418

SCHEMBL13077418

Cc1ocnc1C(=O)N(C)CC(=O)N1CCN(c2ccc(F)cc2C(=O)Nc2nc3c(s2)CN(C)CC3)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.40
ALDH1A1 P00352 3/20 0.40
MAPT P10636 2/20 0.40
F10 P00742 2/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HPGD P15428 2/20 0.40
NPC1 O15118 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
RAB9A P51151 1/20 0.40
LMNA P02545 1/20 0.38
GAA P10253 1/20 0.38
ROCK2 O75116 9/20 0.37
ALOX15 P16050 2/20 0.37
USP2 O75604 1/20 0.37
CASP1 P29466 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL164907 0.90 F10 (0.38) KDM4EALDH1A1MAPTF10KMT2A
SCHEMBL163567 0.90 F10 (0.38) KDM4EALDH1A1MAPTF10KMT2A
SCHEMBL161011 0.76 ALDH1A1 (0.44) KDM4EALDH1A1MAPTF10KMT2A
SCHEMBL13077400 0.75 KDM4E (0.43) KDM4EALDH1A1MAPTF10KMT2A
SCHEMBL112758 0.75 KDM4E (0.42) KDM4EALDH1A1MAPTF10KMT2A
SCHEMBL167393 0.75 KDM4E (0.42) KDM4EALDH1A1MAPTF10KMT2A
SCHEMBL13077016 0.75 CXCR3 (0.47) KDM4EALDH1A1MAPTF10KMT2A
SCHEMBL13077265 0.73 ROCK2 (0.43) KDM4EALDH1A1MAPTF10KMT2A
SCHEMBL112819 0.71 KDM4E (0.39) KDM4EALDH1A1MAPTF10KMT2A
SCHEMBL165338 0.70 CXCR3 (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010126811-A1 CXCR3 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-11-04 WO disclosed