SCHEMBL13085451

SCHEMBL13085451

CCC[C@H](N)C(O)C(F)(F)C(=O)N[C@@H](Cc1ccccc1)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.51
ACE P12821 7/20 0.47
MME P08473 6/20 0.47
ACE2 Q9BYF1 5/20 0.47
REN P00797 1/20 0.46
CPA1 P15085 4/20 0.46
FPR2 P25090 1/20 0.45
ECE1 P42892 1/20 0.45
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
MMP1 P03956 1/20 0.44
MMP3 P08254 1/20 0.44
NAALAD2 Q9Y3Q0 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL464310 0.85 NPSR1 (0.50) NPSR1ACEMMEACE2REN
SCHEMBL12194533 0.80 REN (0.60) NPSR1ACEREN
SCHEMBL13427297 0.79 HDAC3 (0.55) ACEMMEACE2CPA1HDAC3
SCHEMBL13318751 0.76 TACR1 (0.47) ACEREN
SCHEMBL5180357 0.75 NPSR1 (0.69) NPSR1ACEMMEACE2CPA1
SCHEMBL5180354 0.75 NPSR1 (0.69) NPSR1ACEMMEACE2CPA1
SCHEMBL8613833 0.75 NPSR1 (0.69) NPSR1ACEMMEACE2CPA1
SCHEMBL417751 0.74 REN (0.46) ACEMMERENHDAC3HDAC4
Hydrochloric Acid SCHEMBL7348250 0.74 LAP3 (0.44) CPA1
SCHEMBL10408617 0.73 ACE (0.68) NPSR1ACEMMEACE2CPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1878720-B1 Process for preparing chiral bicycloprolinates as intermediates for the preparation of peptidomimetic protease inhibitors VERTEX PHARMA (US) 2010-10-06 EP disclosed