SCHEMBL13088958

SCHEMBL13088958

CC(C)NC(=O)c1cc([N+](=O)[O-])c(SC(C)C2OC(C)O2)cc1C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
SMN1; SMN2 Q16637 4/20 0.38
HTT P42858 3/20 0.38
LMNA P02545 3/20 0.38
CYP3A4 P08684 2/20 0.38
AR P10275 2/20 0.38
GLA P06280 2/20 0.38
CYP1A2 P05177 2/20 0.38
CES2 O00748 1/20 0.38
ABCB11 O95342 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
CHRM1 P11229 1/20 0.38
CYP2C9 P11712 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
TBXA2R P21731 1/20 0.38
AADAC P22760 1/20 0.38
MAPK1 P28482 1/20 0.38
CYP2C19 P33261 1/20 0.38
ADRA1A P35348 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13088890 0.83 HTT (0.37) ALDH1A1SMN1; SMN2HTTLMNACYP3A4
SCHEMBL13088959 0.76 PDGFRB (0.46) ALDH1A1HTTLMNAMEN1KMT2A
SCHEMBL13088964 0.74 TRPA1 (0.47) ALDH1A1SMN1; SMN2HTTLMNACYP3A4
SCHEMBL13089070 0.68 AKR1C3 (0.44) ALDH1A1SMN1; SMN2HTTLMNACYP3A4
SCHEMBL12154447 0.65 AR (0.57) ALDH1A1SMN1; SMN2HTTLMNACYP3A4
SCHEMBL21250383 0.63 HPGD (0.39) ALDH1A1SMN1; SMN2HTTLMNACYP3A4
SCHEMBL12353836 0.63 ALDH1A1 (0.37) ALDH1A1SMN1; SMN2HTTLMNACYP3A4
SCHEMBL2239932 0.61 PDGFRB (0.45) ALDH1A1SMN1; SMN2HTTLMNACYP3A4
SCHEMBL18641484 0.61 MAPT (0.49) ALDH1A1HTTLMNACYP3A4CYP1A2
SCHEMBL13089072 0.60 ALOX5 (0.50) ALDH1A1SMN1; SMN2CYP1A2MAPK1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2243779-A1 BICYCLIC HETEROCYCLIC DERIVATIVE Dainippon Sumitomo Pharma Co., Ltd. (JP) 2010-10-27 EP disclosed