SCHEMBL13093185

SCHEMBL13093185

COC(=O)C1C(c2ccc(F)c(F)c2)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.43
NTRK1 P04629 3/20 0.41
USP30 Q70CQ3 1/20 0.40
NR1H2 P55055 1/20 0.40
NR1H3 Q13133 1/20 0.40
PTPN1 P18031 1/20 0.39
DPP4 P27487 1/20 0.39
GRM5 P41594 2/20 0.39
LMNA P02545 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13093181 0.89 NTRK1 (0.40) PDE4BNTRK1USP30NR1H2NR1H3
SCHEMBL13093170 0.84 SLC6A4 (0.55)
SCHEMBL13092975 0.84 SLC6A4 (0.55)
SCHEMBL13093283 0.84 SLC6A4 (0.55)
SCHEMBL13093189 0.84 SLC6A4 (0.55)
SCHEMBL20806008 0.84 PDE4B (0.42) PDE4BALDH1A1
SCHEMBL5973789 0.84 PDE4B (0.42) PDE4BALDH1A1
SCHEMBL7436099 0.84 PDE4B (0.42) PDE4BALDH1A1
SCHEMBL15185061 0.83 ALDH1A1 (0.50) PDE4BALDH1A1
SCHEMBL16732450 0.82 SLC6A3 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010123006-A1 PYRROLIDINE COMPOUND 武田薬品工業株式会社 (JP) 2010-10-28 WO disclosed