SCHEMBL13136995

SCHEMBL13136995

COc1cccc2c1CC(NCc1ccc(-c3ccc4nc[nH]c4c3)cc1)C2

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.49
ABCB1 P08183 1/20 0.48
QPCT Q16769 11/20 0.41
QPCTL Q9NXS2 6/20 0.41
DRD4 P21917 1/20 0.40
DRD3 P35462 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13137000 0.93 DRD2 (0.53) DRD2ABCB1QPCTDRD4DRD3
SCHEMBL13136998 0.92 DRD2 (0.62) DRD2ABCB1DRD4DRD3
SCHEMBL13136994 0.92 DRD2 (0.62) DRD2ABCB1DRD4DRD3
SCHEMBL13136993 0.89 ABCB1 (0.57) ABCB1QPCTQPCTL
SCHEMBL12634056 0.89 DRD2 (0.48) DRD2QPCTDRD4DRD3
SCHEMBL13136969 0.86 QPCT (0.47) ABCB1QPCTQPCTL
Trifluoroacetic Acid SCHEMBL3052842 0.84 DRD2 (0.44) DRD2ABCB1
Hydrochloric Acid SCHEMBL3047495 0.84 DRD2 (0.52) DRD2ABCB1DRD4DRD3
Hydrochloric Acid SCHEMBL3047492 0.84 DRD2 (0.52) DRD2ABCB1DRD4DRD3
Hydrochloric Acid SCHEMBL3039981 0.83 DRD2 (0.61) DRD2ABCB1DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100222345-A1 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS FOR OPIOID RECEPTORS SMITHKLINE BEECHAM CORPORATION 2010-09-02 US disclosed
US-20100222345-A1 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS FOR OPIOID RECEPTORS SMITHKLINE BEECHAM CORPORATION 2010-09-02 US disclosed
WO-2008021851-A2 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS FOR OPIOID RECEPTORS SMITHKLINE BEECHAM CORPORATION (US) 2008-02-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100222345-A1 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS FOR OPIOID RECEPTORS OPRL1, OPRM1, OPRK1 DRD2 140/4885ABCB1 2258/4885QPCT 1796/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.