SCHEMBL13147201

SCHEMBL13147201

Cc1ccc(-c2ccccc2C(F)(F)F)c(C)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.51
TRPM8 Q7Z2W7 1/20 0.51
TRPV1 Q8NER1 1/20 0.51
S1PR1 P21453 1/20 0.49
HSD11B1 P28845 9/20 0.49
PDK2 Q15119 1/20 0.44
AKR1C3 P42330 1/20 0.42
AKR1C2 P52895 1/20 0.42
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 2/20 0.42
TSHR P16473 2/20 0.42
CYP2C19 P33261 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
CRHR1 P34998 2/20 0.41
ALDH1A1 P00352 2/20 0.41
ELANE P08246 1/20 0.41
LMNA P02545 1/20 0.41
ALOX15 P16050 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22171634 0.89 HSD11B1 (0.50) TRPA1TRPM8TRPV1S1PR1HSD11B1
SCHEMBL278789 0.86 GAA (0.47) TRPA1TRPM8TRPV1S1PR1HSD11B1
SCHEMBL10343225 0.85 TRPA1 (0.51) TRPA1TRPM8TRPV1S1PR1HSD11B1
SCHEMBL26375409 0.85 HSD11B1 (0.50) TRPA1TRPM8TRPV1HSD11B1PDK2
SCHEMBL26262316 0.82 TRPA1 (0.49) TRPA1TRPM8TRPV1S1PR1HSD11B1
SCHEMBL5541462 0.82 HSD11B1 (0.55) TRPA1TRPM8TRPV1S1PR1HSD11B1
SCHEMBL26262326 0.80 TRPA1 (0.47) TRPA1TRPM8TRPV1S1PR1HSD11B1
SCHEMBL23373938 0.79 GAA (0.40) TRPA1TRPM8TRPV1S1PR1HSD11B1
SCHEMBL2600185 0.79 GAA (0.69) PDK2AKR1C3AKR1C2TSHRMEN1
SCHEMBL5964273 0.78 TRPA1 (0.46) TRPA1TRPM8TRPV1S1PR1HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010112461-A1 OXADIAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2010-10-07 WO disclosed