SCHEMBL13147658

SCHEMBL13147658

Cc1cc(-c2cc(N)nc(-c3nc(C(F)(F)F)cs3)n2)c(C)s1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 4/20 0.36
KDM4E B2RXH2 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ALDH1A1 P00352 2/20 0.33
NPC1 O15118 1/20 0.33
MAPT P10636 1/20 0.33
GFER P55789 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PLAU P00749 3/20 0.32
PLA2G10 O15496 1/20 0.32
PTGS2 P35354 1/20 0.32
PTGES O14684 1/20 0.32
C1S P09871 1/20 0.31
TGFBR1 P36897 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.31
HSP90AA1 P07900 1/20 0.31
HSP90AB1 P08238 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL577653 0.88 KDM4E (0.37) IDH1KDM4ESMN1; SMN2ALDH1A1GFER
SCHEMBL13147664 0.86 ALDH1A1 (0.44) IDH1KDM4ESMN1; SMN2ALDH1A1NPC1
SCHEMBL13147662 0.85 IDH1 (0.36) IDH1KDM4ESMN1; SMN2ALDH1A1NPC1
SCHEMBL13147751 0.83 IDH1 (0.36) IDH1PTGESIRAK4HSP90AA1HSP90AB1
SCHEMBL13147748 0.83 IDH1 (0.36) IDH1ALDH1A1NPC1MAPTGFER
SCHEMBL13147740 0.83 IDH1 (0.41) IDH1KDM4EALDH1A1HSD17B10PTGES
SCHEMBL13147672 0.82 SRC (0.38) IDH1ALDH1A1NPC1MAPTGFER
SCHEMBL13147660 0.81 IDH1 (0.39) IDH1KDM4ESMN1; SMN2ALDH1A1NPC1
SCHEMBL13147680 0.81 PTGS2 (0.40) IDH1SMN1; SMN2MAPTPTGS2HSP90AA1
SCHEMBL577580 0.81 IDH1 (0.32) IDH1KDM4ESMN1; SMN2TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118078-A1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARMACEUTICALS, INC. (US) 2010-10-14 WO disclosed