SCHEMBL13147751

SCHEMBL13147751

Cc1cscc1-c1cc(N)nc(-c2nc(C(F)(F)F)cs2)n1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 5/20 0.36
S1PR1 P21453 3/20 0.32
EIF4E P06730 1/20 0.32
PTGES O14684 1/20 0.32
KDM1A O60341 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.31
HSP90AA1 P07900 1/20 0.31
HSP90AB1 P08238 1/20 0.31
SDHB P21912 1/20 0.30
MPL P40238 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL578086 0.86 IDH1 (0.36) IDH1S1PR1EIF4EPTGESIRAK4
SCHEMBL13147658 0.83 IDH1 (0.36) IDH1PTGESIRAK4HSP90AA1HSP90AB1
SCHEMBL13147662 0.83 IDH1 (0.36) IDH1S1PR1PTGESHSP90AA1HSP90AB1
SCHEMBL13147740 0.83 IDH1 (0.41) IDH1PTGESMPL
SCHEMBL13147664 0.81 ALDH1A1 (0.44) IDH1S1PR1HSP90AA1HSP90AB1SDHB
SCHEMBL13147680 0.81 PTGS2 (0.40) IDH1HSP90AA1HSP90AB1
SCHEMBL13147670 0.81 KDM4E (0.36) IDH1HSP90AA1HSP90AB1
SCHEMBL13147748 0.78 IDH1 (0.36) IDH1HSP90AA1HSP90AB1
SCHEMBL577837 0.78 IDH1 (0.33) IDH1S1PR1
SCHEMBL13147742 0.78 IDH1 (0.37) IDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118078-A1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARMACEUTICALS, INC. (US) 2010-10-14 WO disclosed